SCHEMBL762895

SCHEMBL762895

COCCCn1c([C@@H]2CCCN(C(=O)C[C@H](C)Cc3ccc(-c4ccc(S(C)(=O)=O)cc4)cc3)C2)nc2ccccc21

nearest known ligand 0.43

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 10/20 0.43
HRH1 P35367 11/20 0.42
CYP2D6 P10635 7/20 0.42
CHRM1 P11229 3/20 0.41
CYP3A4 P08684 1/20 0.39
PROKR1 Q8TCW9 1/20 0.39
USP2 O75604 1/20 0.38
POLB P06746 1/20 0.38
AGTR1 P30556 1/20 0.38
AGTR2 P50052 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL741301 0.92 HRH1 (0.42) KCNH2HRH1CYP2D6CHRM1CYP3A4
SCHEMBL741300 0.92 HRH1 (0.42) KCNH2HRH1CYP2D6CHRM1CYP3A4
SCHEMBL762888 0.91 KCNH2 (0.45) KCNH2HRH1CYP2D6CHRM1CYP3A4
SCHEMBL762638 0.91 KCNH2 (0.44) KCNH2HRH1CYP2D6CHRM1CYP3A4
SCHEMBL762728 0.89 KCNH2 (0.43) KCNH2HRH1CYP2D6CHRM1CYP3A4
SCHEMBL762721 0.89 KCNH2 (0.46) KCNH2HRH1CYP2D6CHRM1CYP3A4
SCHEMBL762604 0.89 KCNH2 (0.43) KCNH2HRH1CYP2D6CHRM1CYP3A4
SCHEMBL763526 0.89 KCNH2 (0.43) KCNH2HRH1CYP2D6CHRM1CYP3A4
SCHEMBL762619 0.89 KCNH2 (0.43) KCNH2HRH1CYP2D6CHRM1CYP3A4
SCHEMBL762599 0.88 KCNH2 (0.46) KCNH2HRH1CYP2D6CHRM1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed