SCHEMBL763313

SCHEMBL763313

COCCCn1c([C@@H]2CCCN(C(=O)C[C@H](C)Cc3ccc(-c4ccc(C(=O)NCCOC)nc4)cc3)C2)nc2ccccc21

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 10/20 0.41
HRH1 P35367 10/20 0.41
CYP2D6 P10635 7/20 0.41
BTK Q06187 1/20 0.40
CHRM1 P11229 3/20 0.40
CYP3A4 P08684 1/20 0.38
PROKR1 Q8TCW9 1/20 0.37
KDM4E B2RXH2 1/20 0.36
APAF1 O14727 1/20 0.36
USP2 O75604 1/20 0.36
NSD2 O96028 1/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
GLA P06280 1/20 0.36
GAA P10253 1/20 0.36
MAPT P10636 1/20 0.36
HPGD P15428 1/20 0.36
XBP1 P17861 1/20 0.36
CASP1 P29466 1/20 0.36
HTT P42858 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL763307 0.97 KCNH2 (0.41) KCNH2HRH1CYP2D6BTKCHRM1
SCHEMBL739769 0.93 BTK (0.41) KCNH2HRH1CYP2D6BTKCHRM1
SCHEMBL739770 0.93 BTK (0.41) KCNH2HRH1CYP2D6BTKCHRM1
SCHEMBL763542 0.93 KCNH2 (0.42) KCNH2HRH1CYP2D6BTKCHRM1
SCHEMBL763252 0.92 HRH1 (0.44) KCNH2HRH1CYP2D6BTKCHRM1
SCHEMBL740938 0.90 BTK (0.41) KCNH2HRH1CYP2D6BTKCHRM1
SCHEMBL740939 0.90 BTK (0.41) KCNH2HRH1CYP2D6BTKCHRM1
SCHEMBL763506 0.89 KCNH2 (0.44) KCNH2HRH1CYP2D6CHRM1CYP3A4
SCHEMBL765104 0.89 HRH1 (0.38) KCNH2HRH1CYP2D6BTKCHRM1
SCHEMBL744675 0.89 HRH1 (0.40) KCNH2HRH1CYP2D6BTKCHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed