SCHEMBL7637549

SCHEMBL7637549

CCOC(=O)/C=C1/CCC(C)(C)c2cc(C#Cc3ccc(C(=O)OCC)cc3)ccc21

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RARB P10826 13/20 0.48
RARA P10276 10/20 0.48
RARG P13631 10/20 0.48
CYP3A4 P08684 2/20 0.48
KMT2A Q03164 2/20 0.48
CYP26A1 O43174 1/20 0.44
CRABP2 P29373 1/20 0.44
MMP13 P45452 1/20 0.36
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
ESR1 P03372 1/20 0.36
CA7 P43166 1/20 0.36
CA9 Q16790 1/20 0.36
ESR2 Q92731 1/20 0.36
CA14 Q9ULX7 1/20 0.36
ACACB O00763 1/20 0.36
ALDH1A1 P00352 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
NPC1 O15118 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7637556 1.00 RARB (0.48) RARBRARARARGCYP3A4KMT2A
SCHEMBL7641594 0.93 RARB (0.46) RARBRARARARGCYP3A4KMT2A
SCHEMBL7641598 0.93 RARB (0.46) RARBRARARARGCYP3A4KMT2A
SCHEMBL8836952 0.87 RARB (0.50) RARBRARARARGCYP3A4KMT2A
SCHEMBL8836856 0.87 RARB (0.50) RARBRARARARGCYP3A4KMT2A
SCHEMBL5737002 0.85 RARB (0.52) RARBRARARARGCYP3A4KMT2A
SCHEMBL8836693 0.82 RARB (0.49) RARBRARARARGCYP3A4KMT2A
SCHEMBL6293874 0.82 MAPT (0.46) RARBRARARARGCYP3A4KMT2A
SCHEMBL8772609 0.81 RARB (0.48) RARBRARARARGCYP3A4KMT2A
SCHEMBL9484975 0.80 RARB (0.67) RARBRARARARGCYP3A4KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6355806-B1 REGULATORS OF CELL PROLIFERATION AND DIFFERENTIATION, AGENTS FOR TREATING SKIN-RELATED DISEASES ALLERGEN SALES, INC. 2002-03-12 US disclosed
US-5998471-A SKIN DISORDERS; ANTIINFLAMMATORY AGENTS ALLERGAN SALES, INC. (US) 1999-12-07 US disclosed
EP-0800517-A1 ACETYLENES DISUBSTITUTED WITH A 5 OR 8 SUBSTITUTED TETRAHYDRONAPHTHYL OR DIHYDRONAPHTHYL GROUP AND WITH AN ARYL OR HETEROARYL GROUPS HAVING RETINOID-LIKE BIOLOGICAL ACTIVITY Allergan (US) 1997-10-15 EP disclosed
US-5648514-A Substituted acetylenes having retinoid-like biological activity ALLERGAN (US) 1997-07-15 US disclosed
US-5591858-A Acetylenes disubstituted with a 5 substituted tetrahydronaphthyl group and with an aryl or heteroaryl group having retinoid-like biological activity ALLERGAN 1997-01-07 US disclosed
WO-1996020930-A1 ACETYLENES DISUBSTITUTED WITH A 5 OR 8 SUBSTITUTED TETRAHYDRONAPHTHYL OR DIHYDRONAPHTHYL GROUP AND WITH AN ARYL OR HETEROARYL GROUPS HAVING RETINOID-LIKE BIOLOGICAL ACTIVITY ALLERGAN (US) 1996-07-11 WO disclosed