SCHEMBL7646331

SCHEMBL7646331

COc1ccc(N(C)C(=O)NC2C3CCC2CN(CCCNc2ccc(C#N)cc2)C3)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNA5 P22460 1/20 0.40
DRD2 P14416 1/20 0.39
DRD4 P21917 1/20 0.39
DRD3 P35462 1/20 0.39
HRH2 P25021 4/20 0.39
HRH1 P35367 4/20 0.39
CCR6 P51684 1/20 0.39
GRIN2B Q13224 1/20 0.39
HRH3 Q9Y5N1 2/20 0.38
SIRT2 Q8IXJ6 1/20 0.38
GPBAR1 Q8TDU6 1/20 0.37
MCHR1 Q99705 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
CACNA1B Q00975 2/20 0.35
ITK Q08881 2/20 0.35
CCR3 P51677 1/20 0.35
PRKAB2 O43741 1/20 0.35
PRKAG1 P54619 1/20 0.35
PRKAA2 P54646 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7642572 0.86 MCHR1 (0.37) HRH2HRH1HRH3MCHR1CCR3
SCHEMBL7250778 0.83 KCNA5 (0.45) KCNA5DRD2DRD4DRD3HRH2
SCHEMBL7661257 0.82 HRH3 (0.42) KCNA5DRD2DRD4DRD3HRH2
SCHEMBL7246408 0.80 HRH2 (0.41) KCNA5DRD2DRD4DRD3HRH2
SCHEMBL6095849 0.78 GRIN2B (0.61) KCNA5CCR6GRIN2BKMT2A
SCHEMBL7243006 0.75 HRH3 (0.44) HRH2HRH1HRH3MCHR1MEN1
SCHEMBL7252505 0.75 CYP2D6 (0.41) DRD2DRD3HRH2HRH1HRH3
SCHEMBL7242815 0.74 CCR3 (0.41) DRD2DRD3HRH2HRH1HRH3
SCHEMBL7245194 0.73 HRH3 (0.39) KCNA5DRD2DRD4DRD3HRH2
SCHEMBL7248205 0.73 CYP2D6 (0.39) DRD2DRD3HRH2HRH1HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1244631-A1 NEW AZABICYCLOOCTANE DERIVATIVES USEFUL IN THE TREATMENT OF CARDIAC ARRHYTHMIAS AstraZeneca AB (SE) 2002-10-02 EP disclosed
WO-2001047893-A1 NEW AZABICYCLOOCTANE DERIVATIVES USEFUL IN THE TREATMENT OF CARDIAC ARRHYTHMIAS ASTRAZENECA AB (SE) 2001-07-05 WO disclosed