SCHEMBL765033

SCHEMBL765033

Cc1cccc2[nH]c([C@@H]3CCCN(C(=O)C[C@@H](Cc4ccc5ccccc5c4)NC(=O)OC(C)(C)C)C3)nc12

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 0.48
PTGS2 P35354 1/20 0.48
CYP1A2 P05177 4/20 0.41
CYP3A4 P08684 4/20 0.41
CYP2C19 P33261 4/20 0.41
CYP2D6 P10635 3/20 0.41
CYP2C9 P11712 3/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
KDM4E B2RXH2 5/20 0.40
MAPK1 P28482 1/20 0.39
CTSB P07858 1/20 0.39
CTSS P25774 1/20 0.39
CTSK P43235 1/20 0.39
PARP1 P09874 2/20 0.38
TP53 P04637 2/20 0.38
THRB P10828 1/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
HPGD P15428 2/20 0.38
POLB P06746 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10292147 0.92 MAPK1 (0.41) PTGS1PTGS2CYP1A2CYP3A4CYP2C19
SCHEMBL762864 0.85 MAPK1 (0.45) CYP1A2CYP3A4CYP2C19CYP2D6CYP2C9
SCHEMBL762586 0.85 CYP1A2 (0.42) CYP1A2CYP3A4CYP2C19CYP2D6CYP2C9
SCHEMBL762632 0.84 PTGS1 (0.53) PTGS1PTGS2CYP1A2CYP3A4CYP2C19
SCHEMBL763211 0.84 CYP1A2 (0.41) CYP1A2CYP3A4CYP2C19CYP2D6CYP2C9
SCHEMBL762654 0.84 MAPK1 (0.43) CYP1A2CYP3A4CYP2C19CYP2D6CYP2C9
SCHEMBL741843 0.81 PTGS1 (0.51) PTGS1PTGS2CYP1A2CYP3A4CYP2C19
SCHEMBL10293031 0.81 PADI4 (0.38) CYP2D6CTSBCTSSCTSKKMT2A
SCHEMBL762470 0.80 GRIN2B (0.49) CYP1A2CYP3A4CYP2C19CYP2D6CYP2C9
SCHEMBL763367 0.80 GRIN2B (0.49) CYP1A2CYP3A4CYP2C19CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed