SCHEMBL7650657

SCHEMBL7650657

[NH]S(=O)(=O)c1ccc(NN=C2C(=O)Nc3ccc4cn[nH]c4c32)cc1

nearest known ligand 0.35

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
EIF2AK2 P19525 1/20 0.35
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
ALDH1A1 P00352 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7650655 1.00 EIF2AK2 (0.35) EIF2AK2MEN1KMT2AALDH1A1
SCHEMBL5893604 0.89 EIF2AK2 (0.47) EIF2AK2ALDH1A1
SCHEMBL5893613 0.89 EIF2AK2 (0.47) EIF2AK2ALDH1A1
SCHEMBL12856375 0.89 EIF2AK2 (0.47) EIF2AK2ALDH1A1
SCHEMBL7655144 0.75 EIF2AK2 (0.38) EIF2AK2KMT2AALDH1A1
SCHEMBL7655140 0.75 EIF2AK2 (0.38) EIF2AK2KMT2AALDH1A1
SCHEMBL5893496 0.72 EIF2AK2 (0.47) EIF2AK2ALDH1A1
SCHEMBL5893487 0.72 EIF2AK2 (0.47) EIF2AK2ALDH1A1
SCHEMBL6619758 0.72 EIF2AK2 (0.47) EIF2AK2ALDH1A1
SCHEMBL4080527 0.70 CES1 (0.44) MEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6387919-B1 Substituted oxindole derivatives as protein tyrosine kinase and as protein serine/threonine kinase inhibitors GLAXO WELLCOME INC. 2002-05-14 US claimed