SCHEMBL765203

SCHEMBL765203

COCCCn1c([C@@H]2CCCN(C(=O)C[C@H](NC(=O)OC(C)(C)C)c3cccnc3)C2)nc2ccccc21

nearest known ligand 0.42

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 8/20 0.42
ITGA2B P08514 8/20 0.42
KCNH2 Q12809 6/20 0.40
HRH1 P35367 5/20 0.40
CYP2D6 P10635 3/20 0.40
CHRM1 P11229 1/20 0.40
MAPT P10636 2/20 0.36
TP53 P04637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL763828 0.89 KCNH2 (0.43) KCNH2HRH1CYP2D6CHRM1MAPT
SCHEMBL762666 0.89 KCNH2 (0.40) KCNH2HRH1CYP2D6CHRM1MAPT
SCHEMBL763428 0.86 KCNH2 (0.44) KCNH2HRH1CYP2D6CHRM1
SCHEMBL762868 0.86 KCNH2 (0.45) KCNH2HRH1CYP2D6CHRM1
SCHEMBL740472 0.85 KCNH2 (0.45) KCNH2HRH1CYP2D6CHRM1
SCHEMBL741026 0.85 KCNH2 (0.45) KCNH2HRH1CYP2D6CHRM1
SCHEMBL763178 0.82 HRH1 (0.43) KCNH2HRH1CYP2D6CHRM1MAPT
SCHEMBL763858 0.82 KCNH2 (0.42) KCNH2HRH1CYP2D6CHRM1
SCHEMBL762674 0.82 HRH1 (0.41) KCNH2HRH1CYP2D6CHRM1
SCHEMBL763880 0.82 HRH1 (0.43) KCNH2HRH1CYP2D6CHRM1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed