SCHEMBL7652184

SCHEMBL7652184

CS(=O)(=O)OC(=O)c1cc(N)ccc1-c1ccccc1C(=O)Nc1ccc(C(=N)N)cc1

nearest known ligand 0.52

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
F10 P00742 14/20 0.52
F2 P00734 10/20 0.52
PRSS1 P07477 2/20 0.52
PRSS2 P07478 2/20 0.52
PRSS3 P35030 2/20 0.52
F7 P08709 2/20 0.52
F3 P13726 2/20 0.52
PLAU P00749 8/20 0.50
PLAT P00750 8/20 0.50
PLG P00747 4/20 0.50
KLK1 P06870 4/20 0.47
KLK5 Q9Y337 4/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7655173 0.97 F10 (0.49) F10F2PRSS1PRSS2PRSS3
SCHEMBL7663117 0.92 F10 (0.56) F10F2PRSS1PRSS2PRSS3
SCHEMBL7656858 0.90 F10 (0.57) F10F2PRSS1PRSS2PRSS3
SCHEMBL7661924 0.90 F10 (0.55) F10F2PRSS1PRSS2PRSS3
SCHEMBL7663346 0.89 F10 (0.56) F10F2PRSS1PRSS2PRSS3
SCHEMBL7659500 0.89 F10 (0.56) F10F2PRSS1PRSS2PRSS3
SCHEMBL7663676 0.89 F10 (0.52) F10F2PRSS1PRSS2PRSS3
SCHEMBL7663241 0.89 F10 (0.52) F10F2PRSS1PRSS2PRSS3
SCHEMBL7664275 0.89 F10 (0.52) F10F2PRSS1PRSS2PRSS3
SCHEMBL7665826 0.88 F10 (0.61) F10F2PRSS1PRSS2PRSS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6358960-B1 FOR THERAPY OF INTRAVASCULAR COAGULATION, CORONARY THROMBOSIS, CEREBRAL INFARCTION, CEREBRAL EMBOLISM, TRANSIENT ISCHEMIC ATTACK, CEREBROVASCULAR DISORDERS, PULMONARY VASCULAR DISEASES, DEEP VENOUS THROMBOSIS, ETC. ONO PHARMACEUTICAL CO., LTD. (JP) 2002-03-19 US disclosed
EP-1078917-A1 AMIDINO DERIVATIVES AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT ONO PHARMACEUTICAL CO., LTD. (JP) 2001-02-28 EP disclosed