SCHEMBL7652292

SCHEMBL7652292

Cc1cccc(C(=O)O)c1-c1ccccc1C(=O)Nc1ccc(C(=N)N)cc1

nearest known ligand 0.66

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PLAU P00749 6/20 0.66
PLAT P00750 6/20 0.66
F2 P00734 6/20 0.66
F10 P00742 6/20 0.66
KLK1 P06870 6/20 0.66
KLK5 Q9Y337 6/20 0.66
PLG P00747 3/20 0.66
PRSS1 P07477 1/20 0.59
PRSS2 P07478 1/20 0.59
F7 P08709 1/20 0.59
F3 P13726 1/20 0.59
PRSS3 P35030 1/20 0.59
MYC P01106 1/20 0.52
CYP3A4 P08684 1/20 0.51
CYP2C9 P11712 1/20 0.51
ALOX12 P18054 1/20 0.51
GFER P55789 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7655818 0.96 PLAU (0.61) PLAUPLATF2F10KLK1
SCHEMBL7653618 0.95 PLAU (0.66) PLAUPLATF2F10KLK1
SCHEMBL7661225 0.91 F10 (0.61) PLAUPLATF2F10KLK1
SCHEMBL7656724 0.88 PLAU (0.66) PLAUPLATF2F10KLK1
SCHEMBL7658651 0.86 KLK1 (0.67) PLAUPLATF2F10KLK1
SCHEMBL7661930 0.86 CYP3A4 (0.69) PLAUPLATF2F10KLK1
Hydrochloric Acid SCHEMBL7655131 0.85 CYP3A4 (0.68) PLAUPLATF2F10KLK1
SCHEMBL7853538 0.85 PLAU (0.61) PLAUPLATF2F10KLK1
SCHEMBL7855281 0.84 PLAU (0.58) PLAUPLATF2F10KLK1
SCHEMBL7656014 0.84 F10 (0.61) PLAUPLATF2F10KLK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6358960-B1 FOR THERAPY OF INTRAVASCULAR COAGULATION, CORONARY THROMBOSIS, CEREBRAL INFARCTION, CEREBRAL EMBOLISM, TRANSIENT ISCHEMIC ATTACK, CEREBROVASCULAR DISORDERS, PULMONARY VASCULAR DISEASES, DEEP VENOUS THROMBOSIS, ETC. ONO PHARMACEUTICAL CO., LTD. (JP) 2002-03-19 US claimed
EP-1078917-A1 AMIDINO DERIVATIVES AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT ONO PHARMACEUTICAL CO., LTD. (JP) 2001-02-28 EP claimed