SCHEMBL7654293

SCHEMBL7654293

CCCCCCc1cc2c(cc1C#Cc1ccc(CC(=O)O)nn1)C(CC)(CC)CCS2

nearest known ligand 0.31

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 1/20 0.31
CYP3A4 P08684 2/20 0.31
CYP26A1 O43174 1/20 0.31
RARA P10276 1/20 0.31
RARB P10826 1/20 0.31
RARG P13631 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6665619 0.90 CYP3A4 (0.41) PTGDR2CYP3A4CYP26A1RARARARB
SCHEMBL7651542 0.90 CYP3A4 (0.34) CYP3A4CYP26A1RARARARBRARG
SCHEMBL8659725 0.90 CYP3A4 (0.36) CYP3A4RARARARBRARGKMT2A
SCHEMBL7653187 0.88 PTGDR2 (0.35) PTGDR2CYP3A4CYP26A1RARARARB
SCHEMBL7657069 0.86 CYP3A4 (0.37) PTGDR2CYP3A4CYP26A1RARARARB
SCHEMBL7657067 0.86 CYP3A4 (0.35) CYP3A4CYP26A1RARARARBRARG
SCHEMBL7655942 0.85 PTGDR2 (0.31) PTGDR2
SCHEMBL7652220 0.85 CYP3A4 (0.35) CYP3A4RARARARBRARGKMT2A
SCHEMBL8659717 0.82 CYP3A4 (0.31) CYP3A4RARARARBRARGKMT2A
SCHEMBL7652444 0.82 CYP3A4 (0.33) PTGDR2CYP3A4CYP26A1RARARARB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6344463-B1 SKIN DISORDERS, ACNE ALLERGAN SALES, INC. 2002-02-05 US disclosed
EP-0636127-B1 Disubstituted acetylenes bearing heterobicyclic groups and heteroaromatic or phenyl groups having retinoid like activity ALLERGAN INC (US) 2001-04-04 EP disclosed
US-6090826-A Disubstituted acetylenes bearing heterobicyclic groups and heteroaromatic or phenyl groups having retinoid like activity ALLERGAN SALES, INC. (US) 2000-07-18 US disclosed
US-5663347-A REGULATORS OF CELL PROLIFERATION AND DIFFERENTIATION; TREATMENT OF SKIN DISORDERS; ANTICARCINOGNIC AGENTS ALLERGAN (US) 1997-09-02 US disclosed
US-5468879-A Disubstituted acetylenes bearing heterobicyclic groups and heteroaromatic or phenyl groups having retinoid like activity ALLERGAN, INC. (US) 1995-11-21 US disclosed
US-5264578-A Disubstituted acetylenes bearing heterobicyclic groups and heteroaromatic or phenyl groups having retinoid like activity ALLERGAN, INC. (US) 1993-11-23 US disclosed