SCHEMBL7654377

SCHEMBL7654377

CCc1c(N)ccc2c1CN(C(=O)C(F)(F)F)CC2(C)C

nearest known ligand 0.33

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 3/20 0.33
ESR2 Q92731 3/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7649835 0.85 ESR1 (0.34) ESR1ESR2
SCHEMBL7653609 0.84 ESR1 (0.36) ESR1ESR2
SCHEMBL7649698 0.84 ESR1 (0.33) ESR1ESR2
SCHEMBL7655450 0.74 ESR1 (0.42) ESR1ESR2
SCHEMBL7657885 0.74
SCHEMBL18760003 0.71 ESR1 (0.37) ESR1ESR2
SCHEMBL18759901 0.68 ESR1 (0.44) ESR1ESR2
SCHEMBL14348619 0.67 DPP7 (0.43) ESR1ESR2
SCHEMBL30962669 0.67 DPP7 (0.43) ESR1ESR2
SCHEMBL18759982 0.66 ESR1 (0.37) ESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6492378-B1 Substituted isoquinoline derivatives and their use as anticonvulsivants SMITHKLINE BEECHAM P.L.C. (GB) 2002-12-10 US disclosed
EP-1104404-A1 SUBSTITUTED ISOQUINOLINE DERIVATIVES AND THEIR USE AS ANTICONVULSANTS SMITHKLINE BEECHAM PLC (GB) 2001-06-06 EP disclosed
WO-2000009486-A1 SUBSTITUTED ISOQUINOLINE DERIVATIVES AND THEIR USE AS ANTICONVULSIVANTS SMITHKLINE BEECHAM P.L.C. (GB) 2000-02-24 WO disclosed