SCHEMBL7654982

SCHEMBL7654982

CCc1ccc(C(=O)Nc2cc(C)c3c(c2)C(C)(C)N(C)CC3)cc1Br

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.40
RAB9A P51151 4/20 0.40
NPC1 O15118 3/20 0.40
HTR1D P28221 3/20 0.39
HTR1B P28222 3/20 0.39
HTR2A P28223 3/20 0.39
MAPT P10636 4/20 0.39
ALOX15 P16050 1/20 0.39
ALOX12 P18054 1/20 0.39
NR4A1 P22736 1/20 0.39
HSD17B10 Q99714 1/20 0.39
APOBEC3A P31941 1/20 0.36
APOBEC3G Q9HC16 1/20 0.36
MEN1 O00255 5/20 0.36
KMT2A Q03164 5/20 0.36
CYP26A1 O43174 2/20 0.35
CYP3A4 P08684 2/20 0.35
RARA P10276 2/20 0.35
RARB P10826 2/20 0.35
RARG P13631 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7659619 0.99 SMN1; SMN2 (0.39) SMN1; SMN2RAB9ANPC1HTR1DHTR1B
SCHEMBL7655308 0.89 MAPT (0.39) SMN1; SMN2RAB9ANPC1MAPTALOX15
SCHEMBL7653690 0.86 MAPT (0.56) SMN1; SMN2NPC1MAPTALOX15ALOX12
Hydrochloric Acid SCHEMBL7653757 0.85 MAPT (0.55) SMN1; SMN2NPC1MAPTALOX15ALOX12
SCHEMBL7658631 0.85 MAPT (0.45) SMN1; SMN2NPC1HTR1DHTR1BHTR2A
SCHEMBL7653964 0.77 GAA (0.39) SMN1; SMN2RAB9ANPC1MAPTHSD17B10
SCHEMBL7653638 0.76 BRAF (0.47) SMN1; SMN2HTR1DHTR1BHTR2AMAPT
SCHEMBL7660806 0.76 MAPT (0.55) SMN1; SMN2RAB9ANPC1MAPTALOX15
Hydrochloric Acid SCHEMBL7661203 0.76 GAA (0.39) SMN1; SMN2RAB9ANPC1MAPTHSD17B10
Hydrochloric Acid SCHEMBL7662250 0.75 BRAF (0.46) SMN1; SMN2HTR1DHTR1BHTR2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6492378-B1 Substituted isoquinoline derivatives and their use as anticonvulsivants SMITHKLINE BEECHAM P.L.C. (GB) 2002-12-10 US claimed
US-6492378-B1 Substituted isoquinoline derivatives and their use as anticonvulsivants SMITHKLINE BEECHAM P.L.C. (GB) 2002-12-10 US disclosed