SCHEMBL7656740

SCHEMBL7656740

N=C(N)c1ccc(NC(=O)c2cc(Cl)ccc2-c2ccccc2C(=O)OCc2ccccc2)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
F2 P00734 10/20 0.53
F10 P00742 10/20 0.53
PLAU P00749 5/20 0.53
PLAT P00750 5/20 0.53
PLG P00747 5/20 0.53
F7 P08709 7/20 0.51
F3 P13726 7/20 0.51
PRSS1 P07477 1/20 0.51
PRSS2 P07478 1/20 0.51
PRSS3 P35030 1/20 0.51
KLK1 P06870 5/20 0.47
KLK5 Q9Y337 5/20 0.47
PARP1 P09874 1/20 0.45
PARP2 Q9UGN5 1/20 0.45
ALDH1A1 P00352 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7657779 0.91 F10 (0.50) F2F10PLAUPLATPLG
SCHEMBL7658212 0.91 PLAU (0.60) F2F10PLAUPLATPLG
SCHEMBL7654797 0.88 F2 (0.53) F2F10PLAUPLATPLG
SCHEMBL7660778 0.86 F2 (0.55) F2F10PLAUPLATPLG
SCHEMBL7656110 0.86 F2 (0.53) F2F10PLAUPLATPLG
SCHEMBL7656825 0.86 F10 (0.55) F2F10PLAUPLATPLG
SCHEMBL7664302 0.86 F10 (0.57) F2F10PLAUPLATPLG
SCHEMBL7657281 0.85 F10 (0.52) F2F10PLAUPLATPLG
SCHEMBL7664345 0.85 F2 (0.59) F2F10PLAUPLATPLG
SCHEMBL7657027 0.85 F7 (0.61) F2F10PLAUPLATPLG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6358960-B1 FOR THERAPY OF INTRAVASCULAR COAGULATION, CORONARY THROMBOSIS, CEREBRAL INFARCTION, CEREBRAL EMBOLISM, TRANSIENT ISCHEMIC ATTACK, CEREBROVASCULAR DISORDERS, PULMONARY VASCULAR DISEASES, DEEP VENOUS THROMBOSIS, ETC. ONO PHARMACEUTICAL CO., LTD. (JP) 2002-03-19 US disclosed
EP-1078917-A1 AMIDINO DERIVATIVES AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT ONO PHARMACEUTICAL CO., LTD. (JP) 2001-02-28 EP disclosed