SCHEMBL7657511

SCHEMBL7657511

CCn1c(=O)c2[nH]c(C3CCCC3)nc2n2nc(COC(=O)c3ccccc3)nc12

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 3/20 0.49
ADORA1 P30542 11/20 0.48
ADORA2A P29274 5/20 0.48
ADORA2B P29275 3/20 0.48
GMNN O75496 2/20 0.47
LMNA P02545 2/20 0.47
TSHR P16473 2/20 0.47
PMP22 Q01453 2/20 0.47
HIF1A Q16665 2/20 0.47
NPC1 O15118 1/20 0.47
ALDH1A1 P00352 1/20 0.47
TP53 P04637 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2C9 P11712 1/20 0.47
NFKB1 P19838 1/20 0.47
MAPK1 P28482 1/20 0.47
RAB9A P51151 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
HSD17B10 Q99714 1/20 0.47
MEN1 O00255 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6998913 0.86 ADORA1 (0.52) ADORA3ADORA1ADORA2AADORA2BGMNN
SCHEMBL7666412 0.80 ADORA1 (0.51) ADORA3ADORA1ADORA2AADORA2BGMNN
SCHEMBL7662109 0.78 ADORA1 (0.48) ADORA3ADORA1ADORA2AADORA2BGMNN
SCHEMBL7000539 0.78 ADORA1 (0.54) ADORA3ADORA1ADORA2AADORA2BGMNN
SCHEMBL7668320 0.77 ADORA1 (0.53) ADORA3ADORA1ADORA2AADORA2BGMNN
SCHEMBL8567698 0.71 ADORA1 (0.48) ADORA3ADORA1ADORA2AADORA2BGMNN
SCHEMBL8559082 0.65 ADORA1 (0.62) ADORA3ADORA1ADORA2AADORA2BGMNN
SCHEMBL7669969 0.65 ADORA1 (0.40) ADORA3ADORA1ADORA2AADORA2BGMNN
SCHEMBL8561107 0.65 ADORA1 (0.63) ADORA3ADORA1ADORA2AADORA2BGMNN
SCHEMBL7001362 0.64 KMT2A (0.48) ADORA3ADORA1ADORA2AADORA2BLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6492377-B1 Imidazotriazolopyrimidines with adenosine-antagonistic activity BOEHRINGER INGELHEIM PHARMA KG (DE) 2002-12-10 US disclosed