SCHEMBL7658987

SCHEMBL7658987

CCSC1(SCC)CCOc2ccc(C#Cc3ccc(C(CC)CCCC(=O)O)nn3)cc21

nearest known ligand 0.32

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PTGER4 P35408 12/20 0.32
S1PR5 Q9H228 2/20 0.31
CYP3A4 P08684 1/20 0.31
RARA P10276 1/20 0.31
RARB P10826 1/20 0.31
RARG P13631 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7653889 0.80 CYP26A1 (0.36) S1PR5CYP3A4RARARARBRARG
SCHEMBL8662239 0.77 CYP3A4 (0.35) CYP3A4RARARARBRARGKMT2A
SCHEMBL7652437 0.73 CYP3A4 (0.36) PTGER4CYP3A4RARARARBRARG
SCHEMBL7650596 0.72 CYP26A1 (0.39) PTGER4S1PR5CYP3A4RARARARB
SCHEMBL7652315 0.69 CYP26A1 (0.37) S1PR5CYP3A4RARARARBRARG
SCHEMBL7651211 0.69 CYP26A1 (0.37) S1PR5CYP3A4RARARARBRARG
SCHEMBL7652468 0.69 MAP3K14 (0.33)
SCHEMBL6668166 0.69 CYP26A1 (0.46) S1PR5CYP3A4RARARARBRARG
SCHEMBL8662230 0.68 CYP3A4 (0.36) PTGER4CYP3A4RARARARBRARG
SCHEMBL8671496 0.68 KMT2A (0.45) CYP3A4RARARARBRARGKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6344463-B1 SKIN DISORDERS, ACNE ALLERGAN SALES, INC. 2002-02-05 US disclosed
EP-0636127-B1 Disubstituted acetylenes bearing heterobicyclic groups and heteroaromatic or phenyl groups having retinoid like activity ALLERGAN INC (US) 2001-04-04 EP disclosed
US-6090826-A Disubstituted acetylenes bearing heterobicyclic groups and heteroaromatic or phenyl groups having retinoid like activity ALLERGAN SALES, INC. (US) 2000-07-18 US disclosed
US-5663347-A REGULATORS OF CELL PROLIFERATION AND DIFFERENTIATION; TREATMENT OF SKIN DISORDERS; ANTICARCINOGNIC AGENTS ALLERGAN (US) 1997-09-02 US disclosed
US-5468879-A Disubstituted acetylenes bearing heterobicyclic groups and heteroaromatic or phenyl groups having retinoid like activity ALLERGAN, INC. (US) 1995-11-21 US disclosed
EP-0636127-A1 DISUBSTITUTED ACETYLENES BEARING HETEROBICYCLIC GROUPS AND HETEROAROMATIC OR PHENYL GROUPS HAVING RETINOID LIKE ACTIVITY ALLERGAN, INC. (US) 1995-02-01 EP disclosed
US-5264578-A Disubstituted acetylenes bearing heterobicyclic groups and heteroaromatic or phenyl groups having retinoid like activity ALLERGAN, INC. (US) 1993-11-23 US disclosed
WO-1993016068-A1 DISUBSTITUTED ACETYLENES BEARING HETEROBICYCLIC GROUPS AND HETEROAROMATIC OR PHENYL GROUPS HAVING RETINOID LIKE ACTIVITY ALLERGAN, INC. (US) 1993-08-19 WO disclosed