SCHEMBL7659008

SCHEMBL7659008

N=C(N)c1ccc(NC(=O)c2ccccc2-c2ccc(C(=O)OCc3ccccc3)cc2)cc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLAU P00749 4/20 0.62
PLAT P00750 4/20 0.62
F10 P00742 8/20 0.52
F2 P00734 6/20 0.52
GAA P10253 3/20 0.52
PLG P00747 3/20 0.52
KMT2A Q03164 3/20 0.52
RAB9A P51151 2/20 0.52
PRSS1 P07477 3/20 0.52
PRSS2 P07478 3/20 0.52
PRSS3 P35030 3/20 0.52
F7 P08709 3/20 0.52
F3 P13726 3/20 0.52
CHRNB2 P17787 1/20 0.49
CHRNB4 P30926 1/20 0.49
CHRNA3 P32297 1/20 0.49
CHRNA4 P43681 1/20 0.49
KLK1 P06870 6/20 0.48
KLK5 Q9Y337 6/20 0.48
POLB P06746 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7658212 0.90 PLAU (0.60) PLAUPLATF10F2GAA
SCHEMBL7664253 0.90 PLAU (0.61) PLAUPLATF10F2GAA
SCHEMBL7656110 0.84 F2 (0.53) PLAUPLATF10F2PLG
SCHEMBL7660778 0.84 F2 (0.55) PLAUPLATF10F2GAA
SCHEMBL7656825 0.84 F10 (0.55) PLAUPLATF10F2GAA
SCHEMBL7855281 0.84 PLAU (0.58) PLAUPLATF10F2GAA
SCHEMBL7656816 0.84 F2 (0.58) PLAUPLATF10F2GAA
SCHEMBL7664155 0.84 PLAU (0.58) PLAUPLATF10F2PLG
SCHEMBL7657281 0.83 F10 (0.52) PLAUPLATF10F2GAA
SCHEMBL7662830 0.83 PLAU (0.54) PLAUPLATF10F2GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6358960-B1 FOR THERAPY OF INTRAVASCULAR COAGULATION, CORONARY THROMBOSIS, CEREBRAL INFARCTION, CEREBRAL EMBOLISM, TRANSIENT ISCHEMIC ATTACK, CEREBROVASCULAR DISORDERS, PULMONARY VASCULAR DISEASES, DEEP VENOUS THROMBOSIS, ETC. ONO PHARMACEUTICAL CO., LTD. (JP) 2002-03-19 US disclosed
EP-1078917-A1 AMIDINO DERIVATIVES AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT ONO PHARMACEUTICAL CO., LTD. (JP) 2001-02-28 EP disclosed