SCHEMBL765927

SCHEMBL765927

NC(=O)N[C@](Cc1ccccc1)(c1ccc(F)cc1)c1cc(F)cc(OC(F)(F)C(F)F)c1

nearest known ligand 0.60

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CETP P11597 20/20 0.60
KCNH2 Q12809 4/20 0.58
CYP1A2 P05177 1/20 0.52
CYP3A4 P08684 1/20 0.52
CYP2D6 P10635 1/20 0.52
CYP2C9 P11712 1/20 0.52
CYP2C19 P33261 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14533785 0.92 CETP (0.56) CETPKCNH2CYP1A2CYP3A4CYP2D6
SCHEMBL756783 0.89 CETP (0.68) CETPKCNH2
SCHEMBL761468 0.88 CETP (0.58) CETPKCNH2CYP1A2CYP3A4CYP2D6
SCHEMBL758514 0.88 CETP (0.58) CETPKCNH2CYP1A2CYP3A4CYP2D6
SCHEMBL761825 0.88 CETP (0.56) CETPKCNH2CYP1A2CYP3A4CYP2D6
SCHEMBL761826 0.88 CETP (0.56) CETPKCNH2CYP1A2CYP3A4CYP2D6
SCHEMBL758513 0.88 CETP (0.58) CETPKCNH2CYP1A2CYP3A4CYP2D6
SCHEMBL758655 0.88 CETP (0.62) CETPKCNH2
SCHEMBL758720 0.88 CETP (0.62) CETPKCNH2
SCHEMBL758656 0.88 CETP (0.62) CETPKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1954668-B9 HOMO- AND HETEROCYCLIC COMPOUNDS SUITABLE AS CETP INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2012-03-21 EP disclosed
WO-2007062308-A2 HOMO- AND HETEROCYCLIC COMPOUNDS SUITABLE AS CETP INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2007-05-31 WO disclosed