SCHEMBL7663140

SCHEMBL7663140

NS(=O)(=O)c1ccc(CSCc2ccc(CSCc3ccc(CP(=O)(OF)OF)c(Br)c3)cc2)cc1

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 5/20 0.44
CA2 P00918 13/20 0.44
CA1 P00915 10/20 0.44
CA12 O43570 9/20 0.44
CA9 Q16790 9/20 0.44
CA7 P43166 6/20 0.44
CA4 P22748 5/20 0.44
CA5A P35218 5/20 0.44
CA5B Q9Y2D0 5/20 0.44
CA6 P23280 4/20 0.44
CA14 Q9ULX7 4/20 0.44
CA3 P07451 2/20 0.44
CA13 Q8N1Q1 2/20 0.44
NPC1 O15118 1/20 0.34
MAPT P10636 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7595311 0.93 PTPN1 (0.39) PTPN1CA2CA1CA12CA9
SCHEMBL7592239 0.87 PTPN1 (0.50) PTPN1CA2CA1CA12CA9
SCHEMBL7188776 0.86 PTPN1 (0.49) PTPN1CA2CA1CA12CA9
SCHEMBL7595806 0.83 PTPN1 (0.39) PTPN1CA2CA1CA12CA9
SCHEMBL7594100 0.83 PTPN1 (0.48) PTPN1
SCHEMBL7198006 0.82 PTPN1 (0.42) PTPN1MAPT
SCHEMBL7594291 0.81 PTPN1 (0.34) PTPN1
SCHEMBL7594116 0.80 PTPN1 (0.38) PTPN1CA2CA1CA12CA9
SCHEMBL7193468 0.80 PTPN1 (0.45) PTPN1CA2NPC1
SCHEMBL7181995 0.80 PTPN1 (0.37) PTPN1CA2CA1CA12CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6498151-B2 PROTEIN TYROSINE PHOSPHATASES INHIBITORS, ESPECIALLY AS ANTIDIABETIC AGENTS MERCK FROSST CANADA & CO. (CA) 2002-12-24 US claimed