SCHEMBL7685145

SCHEMBL7685145

C=CCN(C)C/C=C/COc1ccc(C(=O)/C=C/C=C(C)C)c(F)c1

nearest known ligand 0.48

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
LSS P48449 13/20 0.48
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
PTPN1 P18031 3/20 0.36
MAOB P27338 3/20 0.35
ALDH1A1 P00352 1/20 0.34
LMNA P02545 1/20 0.34
GAA P10253 1/20 0.34
HPGD P15428 1/20 0.34
ALOX12 P18054 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7685150 1.00 LSS (0.48) LSSMEN1KMT2APTPN1MAOB
Fumaric Acid SCHEMBL7681575 0.97 LSS (0.48) LSSMEN1KMT2APTPN1MAOB
Fumaric Acid SCHEMBL7681568 0.97 LSS (0.48) LSSMEN1KMT2APTPN1MAOB
SCHEMBL7683401 0.85 LSS (0.56) LSSMEN1KMT2AMAOB
SCHEMBL7683408 0.85 LSS (0.56) LSSMEN1KMT2AMAOB
SCHEMBL7688081 0.83 LSS (0.62) LSSPTPN1
SCHEMBL7688083 0.83 LSS (0.62) LSSPTPN1
Fumaric Acid SCHEMBL7688709 0.81 LSS (0.59) LSS
Fumaric Acid SCHEMBL7688712 0.81 LSS (0.59) LSS
SCHEMBL7764135 0.81 MAOB (0.36) MEN1KMT2APTPN1MAOBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6441177-B1 Tertiary amines HOFFMANN-LA ROCHE INC. 2002-08-27 US claimed
EP-0778264-B1 Tertiary amines having antimycotic and cholesterol lowering activity HOFFMANN LA ROCHE (CH) 2001-07-11 EP claimed
EP-0778264-A1 Tertiary amines having antimycotic and cholesterol lowering activity F. HOFFMANN-LA ROCHE AG (CH) 1997-06-11 EP claimed
US-6441177-B1 Tertiary amines HOFFMANN-LA ROCHE INC. 2002-08-27 US disclosed
EP-0778264-B1 Tertiary amines having antimycotic and cholesterol lowering activity HOFFMANN LA ROCHE (CH) 2001-07-11 EP disclosed
US-6034275-A FUGICIDES; ATICHOLESTEROL AGENTS HOFFMANN-LA ROCHE INC. (US) 2000-03-07 US disclosed
EP-0778264-A1 Tertiary amines having antimycotic and cholesterol lowering activity F. HOFFMANN-LA ROCHE AG (CH) 1997-06-11 EP disclosed