SCHEMBL7687433

SCHEMBL7687433

CCNc1c(C)ccnc1Nc1ccc(OCc2ccccc2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 4/20 0.49
ERBB2 P04626 3/20 0.49
AURKB Q96GD4 2/20 0.49
CHEK2 O96017 1/20 0.49
ROS1 P08922 1/20 0.49
FLT3 P36888 1/20 0.49
ERBB4 Q15303 1/20 0.49
CLK4 Q9HAZ1 1/20 0.49
MKNK2 Q9HBH9 1/20 0.49
TTBK1 Q5TCY1 1/20 0.46
TTBK2 Q6IQ55 1/20 0.46
KMT2A Q03164 4/20 0.46
MEN1 O00255 3/20 0.46
MAPT P10636 3/20 0.46
NPC1 O15118 3/20 0.46
RAB9A P51151 3/20 0.46
HPGD P15428 2/20 0.46
TP53 P04637 2/20 0.46
HTT P42858 1/20 0.46
F2 P00734 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7697675 0.84 EGFR (0.46) EGFRERBB2AURKBCHEK2ROS1
SCHEMBL7688389 0.81 EGFR (0.52) EGFRERBB2AURKBCHEK2ROS1
SCHEMBL7688350 0.79 AURKA (0.46) FLT3KMT2AMEN1MAPTHTT
SCHEMBL1699209 0.77 MAPT (0.49) EGFRERBB2AURKBCHEK2ROS1
SCHEMBL6376293 0.76 AR (0.62) KMT2AMEN1MAPTNPC1RAB9A
Hydrochloric Acid SCHEMBL28494253 0.74 AR (0.60) KMT2AMEN1MAPTNPC1RAB9A
SCHEMBL7694335 0.73 EGFR (0.52) EGFRERBB2AURKBCHEK2ROS1
SCHEMBL7694291 0.72 EGFR (0.47) EGFRERBB2AURKBCHEK2ROS1
SCHEMBL7703057 0.72 EGFR (0.55) EGFRERBB2AURKBCHEK2ROS1
SCHEMBL1699142 0.72 EGFR (0.59) EGFRERBB2AURKBCHEK2ROS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011163355-A1 FUSED HETEROCYCLIC COMPOUNDS AS PHOSPHODIESTERASES (PDES) INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2011-12-29 WO disclosed