SCHEMBL7688273

SCHEMBL7688273

O=C(c1ccc(Br)cc1)c1ccc(OCC2CC2CNCC2CC2)cc1F

nearest known ligand 0.67

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
LSS P48449 10/20 0.67
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
PARP10 Q53GL7 2/20 0.43
PARP15 Q460N3 1/20 0.43
KCNH2 Q12809 2/20 0.43
GPR119 Q8TDV5 2/20 0.43
SCN9A Q15858 2/20 0.40
FFAR4 Q5NUL3 1/20 0.38
SRD5A2 P31213 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fumaric Acid SCHEMBL7685404 0.94 LSS (0.61) LSSMEN1KMT2APARP10PARP15
SCHEMBL7687793 0.86 LSS (0.61) LSSMEN1KMT2APARP10PARP15
Hydrochloric Acid SCHEMBL7687465 0.85 LSS (0.60) LSSMEN1KMT2APARP10PARP15
SCHEMBL21123272 0.85 LSS (0.64) LSSMEN1KMT2APARP10PARP15
SCHEMBL7683275 0.82 LSS (0.45) LSSFFAR4
SCHEMBL7681910 0.81 LSS (0.65) LSSMEN1KMT2APARP10PARP15
Fumaric Acid SCHEMBL7687488 0.81 LSS (0.56) LSSPARP10PARP15FFAR4
SCHEMBL17358774 0.80 LSS (1.00) LSSMEN1KMT2APARP10PARP15
SCHEMBL7688275 0.80 LSS (1.00) LSSMEN1KMT2APARP10PARP15
Fumaric Acid SCHEMBL7686200 0.77 LSS (0.42) LSSFFAR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6441177-B1 Tertiary amines HOFFMANN-LA ROCHE INC. 2002-08-27 US claimed
EP-0778264-B1 Tertiary amines having antimycotic and cholesterol lowering activity HOFFMANN LA ROCHE (CH) 2001-07-11 EP claimed
US-6034275-A FUGICIDES; ATICHOLESTEROL AGENTS HOFFMANN-LA ROCHE INC. (US) 2000-03-07 US claimed
US-6441177-B1 Tertiary amines HOFFMANN-LA ROCHE INC. 2002-08-27 US disclosed
US-6034275-A FUGICIDES; ATICHOLESTEROL AGENTS HOFFMANN-LA ROCHE INC. (US) 2000-03-07 US disclosed