SCHEMBL7689050

SCHEMBL7689050

COc1ccc(-c2[nH]c3ccc(OC)c(CCCCCC(=O)N(C)CCCCC(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)F)c3c2C)cc1

nearest known ligand 0.40

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
BCHE P06276 10/20 0.40
ACHE P22303 10/20 0.40
CHRM2 P08172 2/20 0.35
CHRM1 P11229 1/20 0.35
TLR8 Q9NR97 3/20 0.34
TLR7 Q9NYK1 3/20 0.34
TLR9 Q9NR96 2/20 0.34
TACR1 P25103 1/20 0.32
ESR1 P03372 1/20 0.32
ESR2 Q92731 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7688997 0.87 ESR1 (0.46) BCHEACHECHRM2CHRM1TLR8
SCHEMBL7695045 0.86 BCHE (0.37) BCHEACHECHRM2CHRM1TLR8
SCHEMBL8789573 0.79 BCHE (0.38) BCHEACHETLR8TLR7TLR9
SCHEMBL9029036 0.79 TLR9 (0.41) TLR8TLR7TLR9TACR1
SCHEMBL9029025 0.72 FNTA (0.38) TLR8TLR7TLR9TACR1
SCHEMBL9027913 0.72 CCNB2 (0.42) TLR7TLR9TACR1
SCHEMBL7696222 0.72 CCNB2 (0.42) TLR7TLR9TACR1
SCHEMBL9026910 0.69 CCNB2 (0.40) TLR7TLR9TACR1
SCHEMBL8790583 0.69 CCNB2 (0.41) TLR8TLR7TLR9
SCHEMBL8789465 0.68 CCNB2 (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002081444-A1 1-INDOLYL DERIVATIVES, USE THEREOF FOR PRODUCTION OF MEDICAMENTS, A METHOD FOR PRODUCTION OF SAID 1-INDOLYL DERIVATIVES AND PHARMACEUTICAL PREPARATIONS CONTAINING 1-INDOLYL DERIVATIVES SCHERING AKTIENGESELLSCHAFT (DE) 2002-10-17 WO disclosed