SCHEMBL7689993

SCHEMBL7689993

CCN(CC)Cc1ccc(C=Cc2ccccc2C(=O)N[C@@H](Cc2ccccc2)C(=O)CNC(=O)c2ccccc2)cc1

nearest known ligand 0.74

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CAPN1 P07384 14/20 0.74
CTSB P07858 7/20 0.74
CTSS P25774 2/20 0.72
CTSK P43235 2/20 0.72
CTSL P07711 2/20 0.56
PTPN1 P18031 2/20 0.46
BCHE P06276 1/20 0.42
RAB9A P51151 1/20 0.40
HDAC8 Q9BY41 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7688883 0.92 CAPN1 (0.75) CAPN1CTSBCTSSCTSKCTSL
SCHEMBL7696964 0.91 CAPN1 (0.61) CAPN1CTSBCTSSCTSKCTSL
SCHEMBL7690558 0.88 CAPN1 (0.60) CAPN1CTSBCTSSCTSKCTSL
SCHEMBL7691329 0.85 CAPN1 (0.53) CAPN1CTSBCTSSCTSKCTSL
SCHEMBL1335375 0.84 CAPN1 (1.00) CAPN1CTSBCTSSCTSKCTSL
SCHEMBL1335379 0.84 CAPN1 (1.00) CAPN1CTSBCTSSCTSKCTSL
SCHEMBL29483162 0.84 CAPN1 (1.00) CAPN1CTSBCTSSCTSKCTSL
SCHEMBL7690226 0.83 CAPN1 (0.53) CAPN1CTSBCTSSCTSKCTSL
SCHEMBL7688889 0.83 CAPN1 (0.53) CAPN1CTSBCTSSCTSKCTSL
SCHEMBL7696527 0.83 CAPN1 (0.65) CAPN1CTSBCTSSCTSKCTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6436925-B1 BETTER ABLE TO CROSS MEMBRANES; INHIBITORS OF CYSTEINE PROTEASES LIKE CALPAIN I AND II AND CATHEPSIN B AND L, CAN THUS BE USED TO CONTROL DISEASES ASSOCIATED WITH AN ELEVATED ACTIVITY OF CALPAIN ENZYMES OR CATHEPSIN ENZYMES ABBOTT LABORATORIES 2002-08-20 US disclosed