SCHEMBL7693193

SCHEMBL7693193

CC(CNc1ccc([N+](=O)[O-])cc1)Nc1cnc([N+](=O)[O-])c(-c2ccc(Cl)cc2Cl)n1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 1/20 0.44
PIK3CB P42338 1/20 0.44
PIK3CG P48736 1/20 0.44
CRHR1 P34998 1/20 0.42
GSK3B P49841 5/20 0.41
AGPAT2 O15120 1/20 0.38
NPBWR1 P48145 1/20 0.36
MAPT P10636 4/20 0.36
ALDH1A1 P00352 3/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
MEN1 O00255 3/20 0.36
KMT2A Q03164 3/20 0.36
HTT P42858 2/20 0.36
LMNA P02545 2/20 0.36
KDM4E B2RXH2 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA4 P22748 1/20 0.36
CA7 P43166 1/20 0.36
GSK3A P49840 3/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4672350 0.85 GSK3B (0.51) PIK3CAPIK3CBPIK3CGGSK3BAGPAT2
SCHEMBL7084492 0.79 PIK3CA (0.46) PIK3CAPIK3CBPIK3CGGSK3BAGPAT2
SCHEMBL5076249 0.77 GSK3B (0.62) PIK3CAPIK3CBPIK3CGGSK3BNPBWR1
SCHEMBL4670339 0.76 PIK3CA (0.44) PIK3CAPIK3CBPIK3CGGSK3BAGPAT2
SCHEMBL4670338 0.76 GSK3B (0.46) PIK3CAPIK3CBPIK3CGGSK3BNPBWR1
SCHEMBL7084499 0.76 PIK3CA (0.46) PIK3CAPIK3CBPIK3CGCRHR1GSK3B
SCHEMBL4675036 0.75 GSK3B (0.51) PIK3CAPIK3CBPIK3CGCRHR1GSK3B
SCHEMBL4670341 0.74 GSK3B (0.63) PIK3CAPIK3CBPIK3CGCRHR1GSK3B
SCHEMBL7700241 0.73 S1PR4 (0.42) PIK3CAPIK3CBPIK3CGCRHR1GSK3B
SCHEMBL4675353 0.72 GSK3B (0.50) PIK3CAPIK3CBPIK3CGCRHR1GSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001044206-A9 PYRAZINE BASED INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 CHIRON CORP (US) 2002-05-23 WO disclosed