SCHEMBL7696283

SCHEMBL7696283

Cc1cccc(CNC(=O)[C@H]2CC[C@H](Nc3nc4ccccc4[nH]3)CC2)c1

nearest known ligand 0.54

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.54
SMN1; SMN2 Q16637 3/20 0.52
TP53 P04637 1/20 0.49
LPAR2 Q9HBW0 1/20 0.48
NPC1 O15118 2/20 0.47
RAB9A P51151 2/20 0.47
POLB P06746 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
LMNA P02545 4/20 0.46
ITGB3 P05106 1/20 0.43
ITGAV P06756 1/20 0.43
HTT P42858 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7698815 1.00 MAPT (0.54) MAPTSMN1; SMN2TP53LPAR2NPC1
SCHEMBL7696532 0.92 SMN1; SMN2 (0.54) MAPTSMN1; SMN2TP53LPAR2NPC1
SCHEMBL7696529 0.92 SMN1; SMN2 (0.54) MAPTSMN1; SMN2TP53LPAR2NPC1
SCHEMBL7692451 0.89 SMN1; SMN2 (0.55) MAPTSMN1; SMN2TP53NPC1RAB9A
SCHEMBL7698837 0.89 SMN1; SMN2 (0.55) MAPTSMN1; SMN2TP53NPC1RAB9A
SCHEMBL7085647 0.89 SMN1; SMN2 (0.59) MAPTSMN1; SMN2TP53NPC1RAB9A
SCHEMBL7089468 0.89 SMN1; SMN2 (0.59) MAPTSMN1; SMN2TP53NPC1RAB9A
SCHEMBL7085654 0.89 SMN1; SMN2 (0.59) MAPTSMN1; SMN2TP53NPC1RAB9A
SCHEMBL7694033 0.89 SMN1; SMN2 (0.55) MAPTSMN1; SMN2TP53NPC1RAB9A
SCHEMBL7695794 0.89 SMN1; SMN2 (0.52) MAPTSMN1; SMN2TP53NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6291499-B1 TREATING MIGRAINE, DEPRESSION, ANXIETY, SCHIZOPHRENIA, PARKINSON'S DISEASE, OR STROKE MERCK & CO., INC. 2001-09-18 US claimed
US-6495561-B2 TREATING MIGRAINE, DEPRESSION, ANXIETY, SCHIZOPHRENIA, PARKINSON'S DISEASE, OR STROKE MERCK & CO., INC. 2002-12-17 US disclosed
US-6380205-B1 QUINAZOLINE THROUGH A C1-C4ALKYL, C1- C4ALKENYL, C1-C4ALKYNYL, C1-C4ALKOXY, AMINO, AMINOC1-C4ALKYL, HYDROXYC1-C4ALKYL, CARBONYL, CYCLOC3-C6ALKYL OR AMINOCARBONYL CHAIN, USEFUL FOR TREATMENT OF THE PAIN MERCK & CO., INC. 2002-04-30 US disclosed
US-6291499-B1 TREATING MIGRAINE, DEPRESSION, ANXIETY, SCHIZOPHRENIA, PARKINSON'S DISEASE, OR STROKE MERCK & CO., INC. 2001-09-18 US disclosed