SCHEMBL7698804

SCHEMBL7698804

CCCN(CCC)CC(=O)Nc1ccc(-c2n[nH]c3c2Cc2ccccc2-3)cc1

nearest known ligand 0.54

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 13/20 0.54
KDR P35968 4/20 0.53
CDK1 P06493 1/20 0.50
CDK2 P24941 1/20 0.50
KIT P10721 1/20 0.44
FLT1 P17948 1/20 0.44
NPC1 O15118 2/20 0.43
RAB9A P51151 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7698455 0.92 CHEK1 (0.56) CHEK1KDRCDK1CDK2KIT
SCHEMBL7004389 0.89 CHEK1 (0.59) CHEK1KDRNPC1RAB9A
SCHEMBL7095260 0.88 CHEK1 (0.58) CHEK1KDRCDK1CDK2NPC1
SCHEMBL7094049 0.83 CHEK1 (0.60) CHEK1KDRCDK1CDK2NPC1
SCHEMBL7701530 0.83 CHEK1 (0.57) CHEK1KDRCDK1CDK2NPC1
SCHEMBL7092496 0.83 KDR (0.56) CHEK1KDRCDK1CDK2NPC1
SCHEMBL7704050 0.83 CHEK1 (0.52) CHEK1KDRCDK1CDK2NPC1
SCHEMBL7000769 0.82 CHEK1 (0.64) CHEK1KDRCDK1CDK2NPC1
SCHEMBL7704178 0.82 CHEK1 (0.56) CHEK1KDRCDK1CDK2KIT
SCHEMBL7696882 0.82 CHEK1 (0.51) CHEK1KDRCDK1CDK2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6462036-B1 INHIBITING SIGNAL TRANSDUCTION BY MODULATING ACTIVITY OF RECEPTOR AND NONRECEPTOR TYROSINE AND SERINE/THREONINE KINASES TO REGULATE AND MODULATE ABNORMAL OR INAPPROPRIATE CELL PROLIFERATION, DIFFERENTIATION, OR METABOLISM BASF AKTIENGESELLSCHAFT (DE) 2002-10-08 US disclosed