SCHEMBL7699414

SCHEMBL7699414

O=C(NC1CCN(C(=O)N[C@@H](Cc2cc(Br)cc(Br)c2)C(=O)N2CCN(c3ccncc3)CC2)CC1)c1ccccc1

nearest known ligand 0.53

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CALCRL Q16602 17/20 0.53
RAMP1 O60894 9/20 0.53
CALCA P06881 3/20 0.47
POLB P06746 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3965881 1.00 CALCRL (0.53) CALCRLRAMP1CALCAPOLB
SCHEMBL3960149 0.91 CALCRL (0.57) CALCRLRAMP1CALCAPOLB
SCHEMBL3967296 0.86 CALCRL (0.55) CALCRLRAMP1CALCA
SCHEMBL3956564 0.82 CALCRL (0.60) CALCRLRAMP1CALCA
SCHEMBL3965111 0.81 CALCRL (0.62) CALCRLRAMP1CALCA
SCHEMBL3965048 0.81 CALCRL (0.55) CALCRLRAMP1CALCA
SCHEMBL3967290 0.78 CALCRL (0.60) CALCRLRAMP1CALCA
SCHEMBL3954332 0.78 CALCRL (0.82) CALCRLRAMP1CALCA
SCHEMBL3954327 0.78 CALCRL (0.60) CALCRLRAMP1CALCA
SCHEMBL3959858 0.78 CALCRL (0.53) CALCRLRAMP1CALCA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6344449-B1 HEADACHE AND MORPHINE DEPENDENCE DR. KARL THOMAE GMBH (DE) 2002-02-05 US disclosed