SCHEMBL7699569

SCHEMBL7699569

O=C[C@H]1CCO[C@H](OCCc2cc(C(F)(F)F)cc(C(F)(F)F)c2)[C@@H]1c1ccc(F)c(F)c1

nearest known ligand 0.38

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 19/20 0.38
TACR2 P21452 1/20 0.31
TACR3 P29371 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7699574 1.00 TACR1 (0.38) TACR1TACR2TACR3
SCHEMBL7547907 0.90 TACR1 (0.38) TACR1
SCHEMBL7699507 0.90 TACR1 (0.38) TACR1
SCHEMBL6616720 0.90 TACR1 (0.40) TACR1
SCHEMBL6616383 0.90 TACR1 (0.40) TACR1
SCHEMBL6616716 0.90 TACR1 (0.40) TACR1
SCHEMBL7475176 0.87 TACR1 (0.49) TACR1
SCHEMBL7475181 0.87 TACR1 (0.49) TACR1
SCHEMBL7487946 0.87 TACR1 (0.49) TACR1
SCHEMBL6615413 0.80 TACR1 (0.39) TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002016344-A1 TETRAHYDROPYRAN DERIVATIVES AS NK-1 RECEPTOR ANTAGONISTS MERCK SHARP & DOHME LIMITED (GB) 2002-02-28 WO claimed
WO-2002016344-A1 TETRAHYDROPYRAN DERIVATIVES AS NK-1 RECEPTOR ANTAGONISTS MERCK SHARP & DOHME LIMITED (GB) 2002-02-28 WO disclosed