SCHEMBL7700247

SCHEMBL7700247

CCC(Cc1ccc(OC)cc1)=C(c1ccccc1)c1ccc(NCCOC)cc1.CCC(Cc1ccccc1)=C(c1ccccc1)c1ccc(OCCOC)cc1

nearest known ligand 0.52

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 7/20 0.52
CTSS P25774 3/20 0.42
CTSK P43235 3/20 0.42
GCGR P47871 1/20 0.41
KCNH3 Q9ULD8 1/20 0.40
PLAU P00749 1/20 0.40
ELANE P08246 1/20 0.40
PPARG P37231 1/20 0.40
ALDH1A1 P00352 2/20 0.40
MAPT P10636 2/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
RAB9A P51151 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
CTSL P07711 2/20 0.39
CYP19A1 P11511 1/20 0.39
CYP3A4 P08684 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7700245 1.00 ESR1 (0.52) ESR1CTSSCTSKGCGRKCNH3
SCHEMBL7602310 0.94 ESR1 (0.49) ESR1CTSSCTSKKCNH3PLAU
SCHEMBL7602307 0.94 ESR1 (0.49) ESR1CTSSCTSKKCNH3PLAU
SCHEMBL7600070 0.93 ESR1 (0.47) ESR1CTSSCTSKKCNH3PLAU
SCHEMBL7600075 0.93 ESR1 (0.47) ESR1CTSSCTSKKCNH3PLAU
SCHEMBL7602316 0.89 ESR1 (0.53) ESR1CTSSCTSKKCNH3ALDH1A1
SCHEMBL7602320 0.89 ESR1 (0.53) ESR1CTSSCTSKKCNH3ALDH1A1
SCHEMBL7598327 0.88 ESR1 (0.44) ESR1KCNH3ALDH1A1MEN1KMT2A
SCHEMBL7599310 0.88 ESR1 (0.44) ESR1KCNH3ALDH1A1MEN1KMT2A
SCHEMBL7602691 0.86 ESR1 (0.60) ESR1MAPTMEN1KMT2ARAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002066415-A2 NON-STEROIDAL MODULATORS OF ESTROGEN RECEPTORS THE PROVOST, FELLOWS AND SCHOLARS OF THE COLLEGE OF THE HOLY AND UNDIVIDED TRINITY OF QUEEN ELIZABETH NEAR DUBLIN (IE) 2002-08-29 WO disclosed