SCHEMBL7700467

SCHEMBL7700467

CCCN1CCCC(c2nc3c(C(N)=O)cccc3n2CCN2CCCC2)C1

nearest known ligand 0.67

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 12/20 0.67
PARP2 Q9UGN5 1/20 0.53
DRD3 P35462 3/20 0.44
SIGMAR1 Q99720 3/20 0.42
DRD4 P21917 2/20 0.42
NFKB1 P19838 1/20 0.42
PRCP P42785 1/20 0.42
EBP Q15125 1/20 0.42
DRD2 P14416 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5621780 0.99 PARP1 (0.66) PARP1PARP2DRD3SIGMAR1DRD4
SCHEMBL7708434 0.97 PARP1 (0.71) PARP1PARP2DRD3
SCHEMBL5620203 0.96 PARP1 (0.70) PARP1PARP2
SCHEMBL7705470 0.93 PARP1 (0.77) PARP1PARP2
SCHEMBL5621929 0.92 PARP1 (0.64) PARP1PARP2DRD3SIGMAR1DRD4
SCHEMBL5621147 0.92 PARP1 (0.64) PARP1PARP2DRD3SIGMAR1DRD4
SCHEMBL5620536 0.92 PARP1 (0.76) PARP1PARP2
SCHEMBL5621116 0.92 PARP1 (0.67) PARP1PARP2DRD3SIGMAR1DRD4
SCHEMBL5621794 0.90 PARP1 (0.61) PARP1PARP2DRD3SIGMAR1NFKB1
SCHEMBL5621198 0.90 PARP1 (0.61) PARP1PARP2DRD3DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6448271-B1 SUCH AS 2-(PIPERIDIN-4-YL)BENZIMIDAZOLE-4-CARBOXAMIDE; INHIBITORS OF ENZYME POLY(ADP-RIBOSE)POLYMERASE; IMPROVED WATER SOLUBILITY BASF AKTIENGESELLSCHAFT (DE) 2002-09-10 US disclosed