SCHEMBL7700475

SCHEMBL7700475

CCC[C@H]1CC[C@H](N2CCCC(c3nc4cccc(C(N)=O)c4[nH]3)C2)CC1

nearest known ligand 0.50

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 18/20 0.50
PARP2 Q9UGN5 2/20 0.44
POLB P06746 1/20 0.39
BTK Q06187 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7702727 0.95 PARP1 (0.54) PARP1PARP2
SCHEMBL5665661 0.89 PARP1 (0.52) PARP1PARP2
SCHEMBL5622266 0.87 PARP1 (0.62) PARP1PARP2
SCHEMBL5620744 0.86 PARP1 (0.70) PARP1PARP2
SCHEMBL5620739 0.86 PARP1 (0.70) PARP1PARP2
SCHEMBL6781561 0.85 PARP1 (0.50) PARP1PARP2
SCHEMBL5621054 0.82 PARP1 (0.63) PARP1PARP2
SCHEMBL5620556 0.82 PARP1 (0.69) PARP1PARP2
SCHEMBL5621511 0.82 PARP1 (0.70) PARP1PARP2
Hydrochloric Acid SCHEMBL18614332 0.81 PARP1 (0.62) PARP1PARP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6448271-B1 SUCH AS 2-(PIPERIDIN-4-YL)BENZIMIDAZOLE-4-CARBOXAMIDE; INHIBITORS OF ENZYME POLY(ADP-RIBOSE)POLYMERASE; IMPROVED WATER SOLUBILITY BASF AKTIENGESELLSCHAFT (DE) 2002-09-10 US disclosed