SCHEMBL7701206

SCHEMBL7701206

CCN(CC)CCCNC(=O)Nc1ccc(-c2n[nH]c3c2Cc2ccccc2-3)cc1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 11/20 0.49
KDR P35968 3/20 0.48
CDK2 P24941 2/20 0.46
CDK1 P06493 1/20 0.46
ATG4B Q9Y4P1 1/20 0.42
KCNH2 Q12809 1/20 0.41
PDE5A O76074 1/20 0.40
PDE1A P54750 1/20 0.40
PDE1B Q01064 1/20 0.40
PDE3B Q13370 1/20 0.40
PDE1C Q14123 1/20 0.40
PDE3A Q14432 1/20 0.40
CCNE2 O96020 1/20 0.40
CDK4 P11802 1/20 0.40
CCND1 P24385 1/20 0.40
CCNE1 P24864 1/20 0.40
NPC1 O15118 1/20 0.40
PARP1 P09874 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7696838 0.97 CHEK1 (0.48) CHEK1KDRCDK2CDK1ATG4B
SCHEMBL7696882 0.95 CHEK1 (0.51) CHEK1KDRCDK2CDK1KCNH2
SCHEMBL7701117 0.88 CHEK1 (0.51) CHEK1KDRCDK2CDK1KCNH2
SCHEMBL7094461 0.87 CHEK1 (0.56) CHEK1KDRCDK2CDK1ATG4B
SCHEMBL7701963 0.87 CHEK1 (0.57) CHEK1KDRCDK2CDK1KCNH2
SCHEMBL7000883 0.86 KDR (0.55) CHEK1KDRCDK2CDK1NPC1
SCHEMBL7704050 0.84 CHEK1 (0.52) CHEK1KDRCDK2CDK1NPC1
SCHEMBL7698455 0.84 CHEK1 (0.56) CHEK1KDRCDK2CDK1NPC1
SCHEMBL7093375 0.83 CHEK1 (0.50) CHEK1KDRCDK2CDK1NPC1
SCHEMBL6997411 0.82 KDR (0.57) CHEK1KDRCDK2CDK1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6462036-B1 INHIBITING SIGNAL TRANSDUCTION BY MODULATING ACTIVITY OF RECEPTOR AND NONRECEPTOR TYROSINE AND SERINE/THREONINE KINASES TO REGULATE AND MODULATE ABNORMAL OR INAPPROPRIATE CELL PROLIFERATION, DIFFERENTIATION, OR METABOLISM BASF AKTIENGESELLSCHAFT (DE) 2002-10-08 US disclosed