SCHEMBL7701982

SCHEMBL7701982

COC(=O)CN1CCN(CC(OCc2cc(C(F)(F)F)cc(C(F)(F)F)c2)c2ccc(C#N)cc2)CC1

nearest known ligand 0.53

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 12/20 0.53
USP2 O75604 2/20 0.39
CYP2D6 P10635 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
CETP P11597 1/20 0.39
CYP2C19 P33261 1/20 0.39
HTT P42858 1/20 0.37
ELANE P08246 1/20 0.37
TACR2 P21452 1/20 0.37
MEN1 O00255 1/20 0.37
CYP3A4 P08684 1/20 0.37
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7705810 0.90 TACR1 (0.52) TACR1USP2CYP2D6SMN1; SMN2CYP2C19
SCHEMBL7699844 0.88 TACR1 (0.55) TACR1TACR2
SCHEMBL6479244 0.82 TACR1 (0.79) TACR1
SCHEMBL7702022 0.79 TACR1 (0.56) TACR1
SCHEMBL7705392 0.76 TACR1 (0.52) TACR1
SCHEMBL6479302 0.72 TACR1 (0.79) TACR1
SCHEMBL6490118 0.70 TACR1 (0.83) TACR1
SCHEMBL6479029 0.69 TACR1 (1.00) TACR1
SCHEMBL6478575 0.69 TACR1 (0.81) TACR1
SCHEMBL9171577 0.67 POLB (0.59) SMN1; SMN2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1242399-A1 $g(a)-ARYLETHYLPIPERAZINE DERIVATIVES AS NEUROKININ ANTAGONISTS UCB S.A. (BE) 2002-09-25 EP disclosed
WO-2001046167-A1 α-ARYLETHYLPIPERAZINE DERIVATIVES AS NEUROKININ ANTAGONISTS UCB, S.A. (BE) 2001-06-28 WO disclosed