SCHEMBL7702647

SCHEMBL7702647

NC(=O)c1cccc2nc(N3CCCN(CCc4ccc(S(=O)(=O)c5ccccc5)cc4)CC3)[nH]c12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 5/20 0.40
CYP3A4 P08684 1/20 0.39
ABCC1 P33527 1/20 0.39
CASP1 P29466 1/20 0.38
CASP4 P49662 1/20 0.38
CASP5 P51878 1/20 0.38
BTK Q06187 1/20 0.38
CA12 O43570 2/20 0.37
CA1 P00915 2/20 0.37
CA2 P00918 2/20 0.37
CA4 P22748 2/20 0.37
CA5A P35218 2/20 0.37
CA7 P43166 2/20 0.37
CA9 Q16790 2/20 0.37
CA13 Q8N1Q1 2/20 0.37
CA14 Q9ULX7 2/20 0.37
PIK3CA P42336 2/20 0.36
PIM1 P11309 1/20 0.36
FLT3 P36888 1/20 0.36
PIM3 Q86V86 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7702657 0.96 PARP1 (0.42) PARP1CYP3A4ABCC1CASP1CASP4
SCHEMBL7708467 0.87 CYP3A4 (0.42) PARP1CYP3A4ABCC1BTKPIM1
SCHEMBL7702645 0.87 PARP1 (0.52) PARP1PIM1FLT3PIM3BRSK1
SCHEMBL7706393 0.87 CYP3A4 (0.43) PARP1CYP3A4ABCC1BTKHRH1
SCHEMBL7706387 0.87 HRH3 (0.43) PARP1CYP3A4ABCC1BTKAURKB
SCHEMBL7705637 0.87 CYP3A4 (0.41) PARP1CYP3A4ABCC1BTKPIM1
SCHEMBL7700428 0.87 CYP3A4 (0.41) PARP1CYP3A4ABCC1BTKPIM1
SCHEMBL7702571 0.87 CYP3A4 (0.45) PARP1CYP3A4ABCC1BTKCYP2C9
SCHEMBL7700401 0.85 HRH3 (0.48) CYP3A4ABCC1HRH3
SCHEMBL7705476 0.84 HRH3 (0.46) PARP1CYP3A4ABCC1HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6448271-B1 SUCH AS 2-(PIPERIDIN-4-YL)BENZIMIDAZOLE-4-CARBOXAMIDE; INHIBITORS OF ENZYME POLY(ADP-RIBOSE)POLYMERASE; IMPROVED WATER SOLUBILITY BASF AKTIENGESELLSCHAFT (DE) 2002-09-10 US disclosed