SCHEMBL7702652

SCHEMBL7702652

NC(=O)c1cccc2[nH]c(N3CCN(CCc4ccc(S(=O)(=O)c5ccccc5)cc4)CC3)nc12

nearest known ligand 0.55

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 19/20 0.55
PARP2 Q9UGN5 1/20 0.47
AURKA O14965 1/20 0.47
KDR P35968 1/20 0.47
AURKB Q96GD4 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7702645 0.97 PARP1 (0.52) PARP1AURKB
SCHEMBL5620575 0.89 PARP1 (0.51) PARP1PARP2AURKAKDRAURKB
SCHEMBL6872997 0.88 PARP1 (0.41) PARP1
SCHEMBL5621641 0.87 PARP1 (0.61) PARP1AURKAAURKB
SCHEMBL7702657 0.86 PARP1 (0.42) PARP1
SCHEMBL5620008 0.86 PARP1 (0.48) PARP1AURKAAURKB
SCHEMBL5622430 0.86 PARP1 (0.60) PARP1AURKAAURKB
SCHEMBL5622425 0.86 PARP1 (0.64) PARP1AURKAAURKB
SCHEMBL5621272 0.86 PARP1 (0.60) PARP1PARP2AURKAAURKB
SCHEMBL5620669 0.86 PARP1 (0.60) PARP1PARP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6448271-B1 SUCH AS 2-(PIPERIDIN-4-YL)BENZIMIDAZOLE-4-CARBOXAMIDE; INHIBITORS OF ENZYME POLY(ADP-RIBOSE)POLYMERASE; IMPROVED WATER SOLUBILITY BASF AKTIENGESELLSCHAFT (DE) 2002-09-10 US disclosed