SCHEMBL7703602

SCHEMBL7703602

CCN(CC)CC(C)OC(=O)Nc1ccc(-c2n[nH]c3c2Cc2ccccc2-3)cc1

nearest known ligand 0.48

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 11/20 0.48
KDR P35968 4/20 0.47
CDK1 P06493 1/20 0.45
CDK2 P24941 1/20 0.45
SCN1A P35498 1/20 0.40
SCN2A Q99250 1/20 0.40
SCN3A Q9NY46 1/20 0.40
EBP Q15125 1/20 0.40
SIGMAR1 Q99720 1/20 0.40
NPC1 O15118 1/20 0.39
KIT P10721 1/20 0.39
FLT1 P17948 1/20 0.39
HIF1A Q16665 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Acetic Acid SCHEMBL7703507 0.97 KDR (0.47) CHEK1KDRCDK1CDK2SCN1A
SCHEMBL7093375 0.86 CHEK1 (0.50) CHEK1KDRCDK1CDK2NPC1
SCHEMBL7701570 0.85 CHEK1 (0.48) CHEK1KDRCDK1CDK2NPC1
SCHEMBL7698455 0.83 CHEK1 (0.56) CHEK1KDRCDK1CDK2NPC1
SCHEMBL7696867 0.83 CHEK1 (0.47) CHEK1KDRCDK1CDK2NPC1
SCHEMBL7696212 0.83 CHEK1 (0.47) CHEK1KDRCDK1CDK2NPC1
SCHEMBL7814577 0.82 CHEK1 (0.57) CHEK1KDRCDK1CDK2NPC1
SCHEMBL7703509 0.81 CHEK1 (0.46) CHEK1KDRCDK1CDK2SCN1A
Acetic Acid SCHEMBL7696866 0.81 KDR (0.46) CHEK1KDRCDK1CDK2NPC1
SCHEMBL7704050 0.80 CHEK1 (0.52) CHEK1KDRCDK1CDK2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6462036-B1 INHIBITING SIGNAL TRANSDUCTION BY MODULATING ACTIVITY OF RECEPTOR AND NONRECEPTOR TYROSINE AND SERINE/THREONINE KINASES TO REGULATE AND MODULATE ABNORMAL OR INAPPROPRIATE CELL PROLIFERATION, DIFFERENTIATION, OR METABOLISM BASF AKTIENGESELLSCHAFT (DE) 2002-10-08 US disclosed