SCHEMBL7703904

SCHEMBL7703904

CC(C)(Br)c1ccc2c(c1)NC(=O)CC2(C)C

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RARB P10826 1/20 0.48
RARG P13631 1/20 0.48
KIF11 P52732 3/20 0.36
HDAC3 O15379 4/20 0.36
HDAC4 P56524 4/20 0.36
HDAC1 Q13547 4/20 0.36
HDAC2 Q92769 4/20 0.36
HDAC8 Q9BY41 4/20 0.36
HDAC6 Q9UBN7 4/20 0.36
HDAC9 Q9UKV0 4/20 0.36
CMA1 P23946 2/20 0.36
AHR P35869 2/20 0.36
TNKS O95271 1/20 0.33
TNKS2 Q9H2K2 1/20 0.33
TDP2 O95551 2/20 0.33
RXRA P19793 1/20 0.32
RXRB P28702 1/20 0.32
CA9 Q16790 1/20 0.32
EIF2AK2 P19525 1/20 0.32
CRBN Q96SW2 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6578651 0.79 CMA1 (0.59) RARBRARGHDAC3HDAC4HDAC1
SCHEMBL30885057 0.79 CMA1 (0.59) RARBRARGHDAC3HDAC4HDAC1
SCHEMBL11988473 0.77 RARB (0.52) RARBRARGHDAC3HDAC4HDAC1
SCHEMBL14827606 0.76 HDAC3 (0.44) RARBRARGKIF11HDAC3HDAC4
SCHEMBL15577371 0.76 PDK2 (0.50) PGR
SCHEMBL30377238 0.76 CA9 (0.53) RARBRARGHDAC3HDAC4HDAC1
SCHEMBL3140413 0.76 CA9 (0.53) RARBRARGHDAC3HDAC4HDAC1
SCHEMBL9095526 0.76 RARB (0.55) RARBRARGHDAC3HDAC4HDAC1
SCHEMBL6260606 0.76 AHR (0.59) RARBRARGHDAC3HDAC4HDAC1
SCHEMBL6266255 0.76 RARB (0.51) RARBRARGHDAC3HDAC4HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1228042-A2 TETRAHYDROQUINOLINE DERIVATIVES HAVING RETINOID-LIKE BIOLOGICAL ACTIVITY Allergan Sales, Inc. (US) 2002-08-07 EP disclosed
WO-2001012606-A2 TETRAHYDROQUINOLINE DERIVATIVES HAVING RETINOID-LIKE BIOLOGICAL ACTIVITY ALLERGAN SALES, INC. (US) 2001-02-22 WO disclosed