SCHEMBL7704038

SCHEMBL7704038

c1cnc(C2CCOCC2)c(O[C@H]2CCNC2)n1

nearest known ligand 0.52

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7704107 1.00 PDE10A (0.47) PDE10A
Hydrochloric Acid SCHEMBL15134929 0.99 PDE10A (0.46) PDE10A
Hydrochloric Acid SCHEMBL15134930 0.99 PDE10A (0.46) PDE10A
Hydrochloric Acid SCHEMBL15134949 0.99 PDE10A (0.46) PDE10A
SCHEMBL7703048 0.92 PDE10A (0.48) PDE10A
Hydrochloric Acid SCHEMBL15134974 0.90 PDE10A (0.47) PDE10A
SCHEMBL2630958 0.90 PDE10A (0.49) PDE10A
Hydrochloric Acid SCHEMBL15134943 0.89 PDE10A (0.48) PDE10A
SCHEMBL7702975 0.80 PDE10A (0.55) PDE10A
SCHEMBL7702977 0.80 PDE10A (0.55) PDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9376450-B2 Heteroaryloxyheterocyclyl compounds as PDE10 inhibitors AMGEN INC. (US) 2016-06-28 US disclosed
US-9376450-B2 Heteroaryloxyheterocyclyl compounds as PDE10 inhibitors AMGEN INC. (US) 2016-06-28 US disclosed
US-8497265-B2 Heteroaryloxyheterocyclyl compounds as PDE10 inhibitors AMGEN INC. (US) 2013-07-30 US disclosed
US-8497265-B2 Heteroaryloxyheterocyclyl compounds as PDE10 inhibitors AMGEN INC. (US) 2013-07-30 US disclosed
WO-2011143495-A1 HETEROARYLOXYHETEROCYCLYL COMPOUNDS AS PDE10 INHIBITORS AMGEN INC. (US) 2011-11-17 WO disclosed