SCHEMBL7704155

SCHEMBL7704155

CCC(Cc1ccccc1)=C(c1ccccc1)c1ccc(OC(C)N(C)C)cc1.CCC(Cc1ccccc1)=C(c1ccccc1)c1ccc(OC(C)N(CC)CC)cc1.CCC(Cc1ccccc1)=C(c1ccccc1)c1ccc(OC(C)N2CCCC2)cc1.CCC(Cc1ccccc1)=C(c1ccccc1)c1ccc(OC(C)N2CCCCC2)cc1

nearest known ligand 0.46

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 7/20 0.46
ESR2 Q92731 3/20 0.39
PSMB1 P20618 8/20 0.36
PSMB5 P28074 7/20 0.36
PSMB2 P49721 4/20 0.36
LTA4H P09960 1/20 0.34
OPRD1 P41143 1/20 0.34
PDE1A P54750 4/20 0.33
PDE1B Q01064 4/20 0.33
PDE1C Q14123 4/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7603606 0.89 ESR1 (0.55) ESR1ESR2PSMB1PSMB5PSMB2
SCHEMBL7603643 0.89 ESR1 (0.55) ESR1ESR2PSMB1PSMB5PSMB2
SCHEMBL7597044 0.88 ESR1 (0.56) ESR1ESR2PSMB1PSMB5PSMB2
SCHEMBL7597037 0.88 ESR1 (0.56) ESR1ESR2PSMB1PSMB5PSMB2
SCHEMBL7704151 0.86 ESR1 (0.42) ESR1ESR2PSMB1PSMB5PSMB2
SCHEMBL7602287 0.84 ESR1 (0.46) ESR1ESR2PSMB1PSMB5OPRD1
SCHEMBL7602301 0.84 ESR1 (0.46) ESR1ESR2PSMB1PSMB5OPRD1
SCHEMBL7597060 0.83 ESR1 (0.47) ESR1ESR2PSMB1PSMB5OPRD1
SCHEMBL7597047 0.83 ESR1 (0.47) ESR1ESR2PSMB1PSMB5OPRD1
SCHEMBL1962745 0.70 ESR1 (0.59) ESR1ESR2PSMB1PSMB5OPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002066415-A2 NON-STEROIDAL MODULATORS OF ESTROGEN RECEPTORS THE PROVOST, FELLOWS AND SCHOLARS OF THE COLLEGE OF THE HOLY AND UNDIVIDED TRINITY OF QUEEN ELIZABETH NEAR DUBLIN (IE) 2002-08-29 WO claimed