SCHEMBL7705477

SCHEMBL7705477

CCCN1CCN(c2nc3c(C(N)=O)cccc3n2CCN2CCCCC2CC)CC1

nearest known ligand 0.54

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 11/20 0.54
PARP2 Q9UGN5 2/20 0.47
AURKA O14965 2/20 0.41
AURKB Q96GD4 2/20 0.41
ALDH1A1 P00352 2/20 0.40
NPSR1 Q6W5P4 1/20 0.40
THRB P10828 1/20 0.39
LMNA P02545 1/20 0.37
TERT O14746 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5622228 0.97 PARP1 (0.51) PARP1PARP2AURKAAURKBALDH1A1
SCHEMBL7708432 0.89 PARP1 (0.45) PARP1PARP2THRBTERT
SCHEMBL7041918 0.87 PARP1 (0.40) PARP1PARP2ALDH1A1NPSR1THRB
SCHEMBL7700441 0.87 PARP1 (0.58) PARP1PARP2AURKAAURKBALDH1A1
SCHEMBL5619904 0.87 PARP1 (0.67) PARP1PARP2THRBTERT
SCHEMBL7706399 0.86 PARP1 (0.43) PARP1PARP2THRB
SCHEMBL5620118 0.86 PARP1 (0.57) PARP1PARP2AURKAAURKBALDH1A1
SCHEMBL7700394 0.85 PARP1 (0.56) PARP1PARP2AURKAAURKBALDH1A1
SCHEMBL7046250 0.85 PARP1 (0.38) PARP1PARP2ALDH1A1NPSR1THRB
SCHEMBL5621052 0.85 PARP1 (0.55) PARP1PARP2AURKAAURKBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6448271-B1 SUCH AS 2-(PIPERIDIN-4-YL)BENZIMIDAZOLE-4-CARBOXAMIDE; INHIBITORS OF ENZYME POLY(ADP-RIBOSE)POLYMERASE; IMPROVED WATER SOLUBILITY BASF AKTIENGESELLSCHAFT (DE) 2002-09-10 US disclosed