SCHEMBL7706013

SCHEMBL7706013

COC(=O)c1cccc(C=Cc2ccccc2)c1O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 2/20 0.52
CYP1A2 P05177 1/20 0.52
CYP2C19 P33261 1/20 0.52
L3MBTL1 Q9Y468 2/20 0.52
KDM4E B2RXH2 2/20 0.52
BACE1 P56817 1/20 0.52
LMNA P02545 2/20 0.49
TSHR P16473 1/20 0.49
NPC1 O15118 2/20 0.47
RAB9A P51151 2/20 0.47
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
RELA Q04206 1/20 0.47
TRPA1 O75762 2/20 0.46
NFE2L2 Q16236 2/20 0.46
CXCR2 P25025 1/20 0.46
POLB P06746 2/20 0.46
MAPT P10636 3/20 0.44
ALDH1A1 P00352 1/20 0.44
CFTR P13569 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5960456 0.88 CYP1A2 (0.49) HSD17B10CYP1A2CYP2C19L3MBTL1KDM4E
SCHEMBL2658197 0.87 BACE1 (0.61) HSD17B10CYP1A2CYP2C19KDM4EBACE1
SCHEMBL2658196 0.87 BACE1 (0.61) HSD17B10CYP1A2CYP2C19KDM4EBACE1
SCHEMBL29227737 0.87 BACE1 (0.61) HSD17B10CYP1A2CYP2C19KDM4EBACE1
SCHEMBL30423635 0.87 BACE1 (0.61) HSD17B10CYP1A2CYP2C19KDM4EBACE1
SCHEMBL9639720 0.85 HSD17B10 (0.52) HSD17B10CYP1A2CYP2C19L3MBTL1KDM4E
SCHEMBL29627933 0.84 HSD17B10 (0.51) HSD17B10CYP1A2CYP2C19KDM4EBACE1
SCHEMBL29627912 0.84 HSD17B10 (0.51) HSD17B10CYP1A2CYP2C19KDM4EBACE1
SCHEMBL22887320 0.82 PTPN1 (0.57) HSD17B10CYP2C19KDM4ETRPA1MAPT
SCHEMBL7709310 0.82 PTPN1 (0.57) HSD17B10CYP2C19KDM4ETRPA1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104045552-A Medicinal compound as neuroprotective agent SHANGHAI SIMCERE PHARMACEUTICAL RES CO LTD 2014-09-17 CN disclosed
US-6417178-B1 Amyloid binding nitrogen-linked compounds for the antemortem diagnosis of alzheimer's disease, in vivo imaging and prevention of amyloid deposits UNIVERSITY OF PITTSBURGH 2002-07-09 US disclosed
WO-1999024394-A9 COMPOUNDS FOR THE ANTEMORTEM DIAGNOSIS OF ALZHEIMER'S DISEASE AND IN VIVO IMAGING AND PREVENTION OF AMYLOID DEPOSITION UNIV PITTSBURGH (US) 2001-05-31 WO disclosed
EP-1028941-A2 COMPOUNDS FOR THE ANTEMORTEM DIAGNOSIS OF ALZHEIMER'S DISEASE AND IN VIVO IMAGING AND PREVENTION OF AMYLOID DEPOSITION UNIVERSITY OF PITTSBURGH (US) 2000-08-23 EP disclosed
WO-1999024394-A2 COMPOUNDS FOR THE ANTEMORTEM DIAGNOSIS OF ALZHEIMER'S DISEASE AND IN VIVO IMAGING AND PREVENTION OF AMYLOID DEPOSITION UNIVERSITY OF PITTSBURGH (US) 1999-05-20 WO disclosed