SCHEMBL7706494

SCHEMBL7706494

CC(=O)Nc1ccc(Sc2ccc(C(=O)N[C@@H]3C4CCN(CC4)[C@H]3C)cc2)s1.CC(=O)c1ccc(Sc2ccc(C(=O)N[C@@H]3C4CCN(CC4)[C@H]3C)cc2)s1

nearest known ligand 0.39

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 12/20 0.39
CHRNB2 P17787 11/20 0.35
CHRNA4 P43681 11/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6874983 0.95 CHRNA7 (0.42) CHRNA7CHRNB2CHRNA4
SCHEMBL6882136 0.93 CHRNA7 (0.42) CHRNA7CHRNB2CHRNA4
SCHEMBL7063154 0.85 CHRNA7 (0.38) CHRNA7CHRNB2CHRNA4
SCHEMBL7061872 0.84 CHRNA7 (0.39) CHRNA7CHRNB2CHRNA4
SCHEMBL6884781 0.81 CHRNA7 (0.43) CHRNA7CHRNB2CHRNA4
SCHEMBL7063330 0.81 CHRNA7 (0.38) CHRNA7CHRNB2CHRNA4
SCHEMBL6875498 0.80 CHRNA7 (0.42) CHRNA7CHRNB2CHRNA4
SCHEMBL7064115 0.80 CHRNA7 (0.40) CHRNA7CHRNB2CHRNA4
SCHEMBL6882726 0.80 ITK (0.46) CHRNA7
SCHEMBL6882524 0.80 CHRNA7 (0.47) CHRNA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6486172-B2 ADMINISTERING TO A MAMMAL A THERAPEUTICALLY EFFECTIVE AMOUNT OF BENZAMIDE OR BENZOCARBONYLSULFIDE SUBSTITUTED 1-AZABICYCLO(2,2,2)OCT-3-YL COMPOUNDS TO TREAT THE CONDITIONS ASSOCIATED WITH DEFECTS OF NICOTINIC SUBTYPES BRAIN RECEPTORS PHARMACIA & UPJOHN COMPANY 2002-11-26 US claimed