SCHEMBL7706677

SCHEMBL7706677

COC#Cc1cccc(C#N)c1

nearest known ligand 0.53

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 3/20 0.45
ENPP2 Q13822 1/20 0.41
AR P10275 1/20 0.41
FFAR1 O14842 1/20 0.41
TSHR P16473 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30873480 0.80 GRM5 (0.55) GRM5ENPP2FFAR1TSHR
Charcoal, Activated SCHEMBL31286316 0.78 GRM5 (0.53) GRM5ENPP2FFAR1TSHR
SCHEMBL9289 0.78 TSHR (0.61) GRM5ENPP2TSHR
SCHEMBL2817154 0.78 TSHR (0.61) GRM5ENPP2TSHR
Water SCHEMBL28137572 0.78 TSHR (0.61) GRM5ENPP2TSHR
SCHEMBL22431368 0.77 GRM5 (0.49) GRM5ENPP2FFAR1TSHR
SCHEMBL27916593 0.76 GRM5 (0.54) GRM5FFAR1
SCHEMBL1745083 0.76 GRM5 (0.33) GRM5
Hydrochloric Acid SCHEMBL19327577 0.75 TSHR (0.58) GRM5ENPP2TSHR
Fluoride SCHEMBL28362409 0.75 TSHR (0.58) GRM5ENPP2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6355490-B1 CODING INDIVIDUAL MEMBERS OF LIBRARY; COVALENTLY BONDING NITRILE TO SOLID SUPPORT; DETECTION BY INFRARED OR RAMAN SPECTROSCOPY ABBOTT LABORATORIES 2002-03-12 US disclosed
US-6274385-B1 COVALENTLY ATTACHING TO EACH SOLID SUPPORT AT LEAST ONE ACETYLENE CODING IDENTIFIER DETECTABLE BY INFRARED OR RAMAN SPECTROSCOPY TO CODE INDIVIDUAL MEMBERS OF A COMBINATORIAL CHEMICAL LIBRARY ABBOTT LABORATORIES 2001-08-14 US disclosed
EP-0879219-B1 ATTACHED TAGS FOR USE IN COMBINATORIAL CHEMISTRY SYNTHESIS ABBOTT LAB (US) 2000-03-01 EP disclosed
EP-0879219-A1 ATTACHED TAGS FOR USE IN COMBINATORIAL CHEMISTRY SYNTHESIS Abbott Laboratories (US) 1998-11-25 EP disclosed
WO-1998011036-A9 ATTACHED TAGS FOR USE IN COMBINATORIAL CHEMISTRY SYNTHESIS 1998-07-09 WO disclosed
WO-1998011036-A1 ATTACHED TAGS FOR USE IN COMBINATORIAL CHEMISTRY SYNTHESIS ABBOTT LABORATORIES (US) 1998-03-19 WO disclosed