SCHEMBL7709212

SCHEMBL7709212

COc1ccc(-c2cc(N)n3nc(-c4ccccn4)nc3c2)cc1OC

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 1/20 0.49
KLK3 P07288 1/20 0.47
CSNK1D P48730 1/20 0.47
KDM4E B2RXH2 1/20 0.47
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
DCTPP1 Q9H773 1/20 0.47
ATM Q13315 5/20 0.45
PIK3CA P42336 1/20 0.45
PIK3CB P42338 1/20 0.45
MTOR P42345 1/20 0.45
PRKDC P78527 1/20 0.45
POLB P06746 1/20 0.44
MAPT P10636 2/20 0.42
ALDH1A1 P00352 2/20 0.42
NPC1 O15118 1/20 0.42
TUBB4A P04350 1/20 0.42
TUBB P07437 1/20 0.42
TUBA3C P0DPH7 1/20 0.42
TUBA1B P68363 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7431382 0.87 NPC1 (0.52) ADORA2AKDM4EMEN1KMT2ADCTPP1
SCHEMBL7709217 0.86 GRM5 (0.50) ADORA2AKLK3KDM4EDCTPP1ATM
SCHEMBL7483006 0.85 NPC1 (0.53) ADORA2AKDM4EMEN1KMT2ADCTPP1
SCHEMBL7708845 0.83 ADORA2A (0.54) ADORA2AKDM4EMEN1KMT2ADCTPP1
SCHEMBL7428533 0.82 ADORA2A (0.60) ADORA2AKDM4EMEN1KMT2AMAPT
SCHEMBL7703002 0.82 ADORA2A (0.47) ADORA2AKDM4EMEN1KMT2AATM
SCHEMBL7481790 0.81 ADORA2A (0.52) ADORA2AKDM4EMEN1KMT2AMAPT
SCHEMBL7709146 0.81 ADORA2A (0.52) ADORA2AKDM4EMEN1KMT2ADCTPP1
SCHEMBL7708907 0.81 ADORA2A (0.52) ADORA2AKDM4EMEN1KMT2AMAPT
SCHEMBL7427435 0.81 ADORA2A (0.54) ADORA2AKDM4EMEN1KMT2ADCTPP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6355653-B1 DRUG AND CARRIER FOR ANTIALLERGENS, BRAIN DISORDERS AND NEUROTRANSMITTERS HOFFMANN-LA ROCHE INC. 2002-03-12 US disclosed