SCHEMBL7709370

SCHEMBL7709370

COc1cc2c3c(ccc(C)c3c1NC(C)=O)C(=O)N(O)C2=O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.44
KMT2A Q03164 4/20 0.44
KDM4E B2RXH2 3/20 0.44
MAPT P10636 3/20 0.44
POLB P06746 2/20 0.44
LMNA P02545 1/20 0.44
PABPC1 P11940 1/20 0.44
XBP1 P17861 1/20 0.44
NFKB1 P19838 1/20 0.44
HTT P42858 1/20 0.44
SMARCA2 P51531 1/20 0.44
NFKB2 Q00653 1/20 0.44
RELA Q04206 1/20 0.44
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
ADORA3 P0DMS8 4/20 0.37
ADORA2A P29274 1/20 0.37
ADORA2B P29275 1/20 0.37
HSD17B10 Q99714 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7712139 0.84 NPC1 (0.41) ALDH1A1KMT2AKDM4EMAPTPOLB
SCHEMBL7709779 0.69 MAPT (0.50) ALDH1A1KMT2AKDM4EMAPTPOLB
SCHEMBL3285076 0.67 CA1 (0.52) ALDH1A1KMT2AKDM4EMAPTPOLB
SCHEMBL7709368 0.66 MAPT (0.56) ALDH1A1KMT2AKDM4EMAPTPOLB
SCHEMBL10683659 0.66 HSD17B10 (0.47) ALDH1A1KMT2AKDM4EMAPTHSD17B10
SCHEMBL1025411 0.64 ERCC1 (0.62) ALDH1A1KMT2AKDM4EMAPTPOLB
SCHEMBL7712214 0.64 MAPT (0.71) ALDH1A1KMT2AKDM4EMAPTPOLB
SCHEMBL7712200 0.64 KMT2A (0.50) ALDH1A1KMT2AKDM4EMAPTPOLB
SCHEMBL2633374 0.64 PRMT1 (0.59) ALDH1A1KMT2AKDM4EMAPTPOLB
SCHEMBL7709776 0.63 KLK7 (0.53) ALDH1A1KMT2AKDM4EMAPTPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6362181-B1 BACTERICIDES; ENZYME INHIBITORS; ANTITUMOR AGENTS WARNER-LAMBERT COMPANY 2002-03-26 US claimed
US-6362181-B1 BACTERICIDES; ENZYME INHIBITORS; ANTITUMOR AGENTS WARNER-LAMBERT COMPANY 2002-03-26 US disclosed
US-6177423-B1 N-(HYDROXY OR PROTECTED HYDROXY)-BENZO(DE)ISOQUINOLINE-1,3-DIONE DERIVATIVES; BACTERIAL DNA GYRASE AND DNA TOPOISOMERASE INHIBITORS USEFUL FOR ANTIBACTERIAL AGENTS HAVING REDUCED DRUG RESISTANCE AND REDUCED SIDE EFFECTS WARNER-LAMBERT COMPANY 2001-01-23 US disclosed