SCHEMBL7709537

SCHEMBL7709537

O=C1OC(=O)c2cc(F)c(O)c3cccc1c23

nearest known ligand 0.49

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
TYMS P04818 7/20 0.49
NMUR2 Q9GZQ4 2/20 0.39
ALOX15 P16050 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
DHFR P00374 2/20 0.37
AHR P35869 1/20 0.35
ERN1 O75460 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7709692 0.86 TYMS (0.51) TYMSALOX15TDP1DHFR
SCHEMBL29836499 0.80 TYMS (0.49) TYMSALOX15TDP1
SCHEMBL4959190 0.77 TYMS (0.61) TYMSALOX15TDP1DHFRAHR
SCHEMBL7709648 0.76 TYMS (0.45) TYMSALOX15TDP1
SCHEMBL7703859 0.73 TYMS (0.49) TYMSALOX15TDP1DHFR
SCHEMBL30608351 0.73 TYMS (0.61) TYMSALOX15TDP1
SCHEMBL4533766 0.73 TYMS (0.61) TYMSALOX15TDP1
SCHEMBL10267341 0.72 TYMS (0.70) TYMSALOX15TDP1
SCHEMBL6719946 0.72 TYMS (0.55) TYMSALOX15TDP1
SCHEMBL9078978 0.71 TYMS (0.46) TYMSALOX15TDP1AHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6362181-B1 BACTERICIDES; ENZYME INHIBITORS; ANTITUMOR AGENTS WARNER-LAMBERT COMPANY 2002-03-26 US disclosed
US-6177423-B1 N-(HYDROXY OR PROTECTED HYDROXY)-BENZO(DE)ISOQUINOLINE-1,3-DIONE DERIVATIVES; BACTERIAL DNA GYRASE AND DNA TOPOISOMERASE INHIBITORS USEFUL FOR ANTIBACTERIAL AGENTS HAVING REDUCED DRUG RESISTANCE AND REDUCED SIDE EFFECTS WARNER-LAMBERT COMPANY 2001-01-23 US disclosed
EP-0939754-A2 N-OXY-NAPHTHALIMIDES AS ANTIBACTERIAL AGENTS WARNER-LAMBERT COMPANY (US) 1999-09-08 EP disclosed
WO-1998019648-A2 N-OXY-NAPHTHALIMIDES AS ANTIBACTERIAL AGENTS WARNER-LAMBERT COMPANY (US) 1998-05-14 WO disclosed