SCHEMBL7709642

SCHEMBL7709642

CC(=O)c1ccc2cccc3c2c1C(=O)OC3=O

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TYMS P04818 8/20 0.55
HSD17B10 Q99714 3/20 0.42
KDM4E B2RXH2 3/20 0.42
ALDH1A1 P00352 3/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
HPGD P15428 2/20 0.42
NPSR1 Q6W5P4 1/20 0.40
MAOB P27338 3/20 0.38
PDK2 Q15119 1/20 0.38
MAOA P21397 1/20 0.38
CYP1A2 P05177 2/20 0.36
CA12 O43570 1/20 0.36
NT5E P21589 1/20 0.36
CA9 Q16790 1/20 0.36
CES2 O00748 1/20 0.36
BCHE P06276 1/20 0.36
CES1 P23141 1/20 0.36
MCL1 Q07820 1/20 0.36
CYP2C19 P33261 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18301594 0.80 PDK2 (0.44) TYMSALDH1A1MEN1KMT2AMAOB
SCHEMBL1667013 0.78 KMT2A (0.41) TYMSHSD17B10KDM4EALDH1A1MEN1
SCHEMBL1052126 0.77 PARP1 (0.56) TYMSHSD17B10KDM4EALDH1A1MEN1
SCHEMBL7750777 0.77 TYMS (0.62) TYMSHSD17B10KDM4EALDH1A1MEN1
SCHEMBL7841346 0.76 TYMS (0.73) TYMSKDM4EALDH1A1MEN1KMT2A
SCHEMBL13069937 0.74 TYMS (0.51) TYMSKDM4EALDH1A1MEN1KMT2A
SCHEMBL28272717 0.74 TYMS (0.58) TYMSHSD17B10KDM4EALDH1A1MEN1
SCHEMBL1517949 0.74 TYMS (0.46) TYMSKDM4EALDH1A1MEN1KMT2A
SCHEMBL4960210 0.73 TYMS (0.62) TYMSHSD17B10KDM4EALDH1A1HPGD
SCHEMBL22580735 0.73 TYMS (0.62) TYMSHSD17B10KDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6362181-B1 BACTERICIDES; ENZYME INHIBITORS; ANTITUMOR AGENTS WARNER-LAMBERT COMPANY 2002-03-26 US disclosed
US-6177423-B1 N-(HYDROXY OR PROTECTED HYDROXY)-BENZO(DE)ISOQUINOLINE-1,3-DIONE DERIVATIVES; BACTERIAL DNA GYRASE AND DNA TOPOISOMERASE INHIBITORS USEFUL FOR ANTIBACTERIAL AGENTS HAVING REDUCED DRUG RESISTANCE AND REDUCED SIDE EFFECTS WARNER-LAMBERT COMPANY 2001-01-23 US disclosed
EP-0939754-A2 N-OXY-NAPHTHALIMIDES AS ANTIBACTERIAL AGENTS WARNER-LAMBERT COMPANY (US) 1999-09-08 EP disclosed
WO-1998019648-A2 N-OXY-NAPHTHALIMIDES AS ANTIBACTERIAL AGENTS WARNER-LAMBERT COMPANY (US) 1998-05-14 WO disclosed