SCHEMBL7710771

SCHEMBL7710771

CC1Oc2ccc(-c3cccs3)cc2NC1=S

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.41
SLC6A11 P48066 1/20 0.40
PGR P06401 2/20 0.40
PDE3B Q13370 2/20 0.36
PDE3A Q14432 2/20 0.36
LPL P06858 1/20 0.36
LIPG Q9Y5X9 1/20 0.36
ALOX5 P09917 2/20 0.33
PARP1 P09874 2/20 0.33
KDR P35968 1/20 0.33
ERN1 O75460 1/20 0.33
PTGS1 P23219 1/20 0.33
PTGS2 P35354 1/20 0.33
HTR1D P28221 1/20 0.33
HTR1B P28222 1/20 0.33
PRMT6 Q96LA8 1/20 0.33
HDAC3 O15379 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC2 Q92769 1/20 0.33
PDK2 Q15119 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7000241 0.84 PARP1 (0.52) KCNH2SLC6A11PGRPDE3BPDE3A
SCHEMBL7000985 0.79 KDM4E (0.54) PGRPDE3BPDE3APARP1KDM4E
SCHEMBL7711118 0.77 KCNH2 (0.40) KCNH2PGRPDE3BPDE3ALPL
SCHEMBL7711311 0.73 CYP11B1 (0.48) PDE3BPDE3AKDR
SCHEMBL7988135 0.72 BRD4 (0.53) PARP1MEN1GAAKMT2A
SCHEMBL7711230 0.71 PARP1 (0.37) PDE3BPDE3APARP1
SCHEMBL7000474 0.71 PARP1 (0.37) PDE3BPDE3APARP1KDM4EMEN1
SCHEMBL6998842 0.71 ACE2 (0.40) PARP1PTGS1PTGS2KDM4EMEN1
SCHEMBL7003121 0.70 KCNH2 (0.46) KCNH2SLC6A11PGRLPLLIPG
SCHEMBL7003125 0.68 KCNH2 (0.48) KCNH2PGRHDAC3HDAC1HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6365736-B1 TREATMENT OF NERVOUS SYSTEM DISORDERS, CARDIOVASCULAR DISORDERS AND FOR ACTIVITY AS NO-SYNTHASES (NOS) INHIBITORS. SCHERING AKTIENGESELLSCHAFT (DE) 2002-04-02 US disclosed