SCHEMBL7713293

SCHEMBL7713293

CC(=O)OCc1cn(C(c2ccccc2)(c2ccccc2)c2ccccc2)c(-c2nc(CO)cn2C(c2ccccc2)(c2ccccc2)c2ccccc2)n1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.40
ACSS2 Q9NR19 1/20 0.38
CYP1A2 P05177 2/20 0.35
CYP2C19 P33261 2/20 0.35
TSHR P16473 3/20 0.35
NPC1 O15118 2/20 0.34
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
CYP2C9 P11712 1/20 0.33
ELANE P08246 1/20 0.33
POLB P06746 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
OPRM1 P35372 1/20 0.33
OPRD1 P41143 1/20 0.33
IDH1 O75874 1/20 0.32
SIRT2 Q8IXJ6 3/20 0.32
MAPK1 P28482 1/20 0.32
TP53 P04637 1/20 0.32
PKM P14618 1/20 0.32
NFKB1 P19838 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7939502 0.81 BACE1 (0.33) ALDH1A1NPC1RAB9ASMN1; SMN2
SCHEMBL10676751 0.76 NOTUM (0.36) ALDH1A1ACSS2TSHRMEN1KMT2A
SCHEMBL7713289 0.76 SIRT2 (0.46) ALDH1A1NPC1SIRT2
SCHEMBL10917397 0.73 NOTUM (0.39) L3MBTL1
SCHEMBL3573464 0.72 SIRT2 (0.49) ALDH1A1CYP1A2CYP2C19NPC1MEN1
SCHEMBL17651946 0.72 MAPK1 (0.35) ALDH1A1MEN1KMT2AL3MBTL1MAPK1
Alcohol SCHEMBL6432975 0.72 SIRT2 (0.47) ALDH1A1NPC1SIRT2
SCHEMBL6971146 0.71 KDM4E (0.37) ALDH1A1MEN1KMT2APOLBOPRM1
SCHEMBL8022922 0.70 NOTUM (0.36) L3MBTL1
SCHEMBL10916083 0.70 CYP2J2 (0.37) ALDH1A1ACSS2CYP1A2CYP2C19NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1214326-A1 INHIBITORS OF PRENYL-PROTEIN TRANSFERASE Merck & Co., Inc. (US) 2002-06-19 EP disclosed
WO-2001018006-A1 INHIBITORS OF PRENYL-PROTEIN TRANSFERASE MERCK & CO., INC. (US) 2001-03-15 WO disclosed