SCHEMBL7720296

SCHEMBL7720296

COc1ccc2ccc(C#N)cc2c1C(C)=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA9 Q16790 1/20 0.46
NCEH1 Q6PIU2 3/20 0.43
AR P10275 3/20 0.41
ALDH1A1 P00352 2/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
GAA P10253 2/20 0.38
MMP3 P08254 1/20 0.38
PDE4A P27815 1/20 0.38
PDE4B Q07343 1/20 0.38
PDE4C Q08493 1/20 0.38
PDE4D Q08499 1/20 0.38
MAPK1 P28482 1/20 0.38
MAPT P10636 2/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
USP2 O75604 1/20 0.38
MCL1 Q07820 1/20 0.38
P4HB P07237 1/20 0.38
PDE5A O76074 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7725096 0.85 AR (0.41) NCEH1ARALDH1A1CA1CA2
SCHEMBL7344856 0.78 AR (0.45) NCEH1ARCA1CA2MCL1
SCHEMBL20855586 0.76 AR (0.50) CA9ARALDH1A1GAAPDE4A
SCHEMBL30468153 0.76 AR (0.50) CA9ARALDH1A1GAAPDE4A
SCHEMBL7723749 0.76 AR (0.50) NCEH1ARALDH1A1CA1CA2
SCHEMBL7337530 0.76 AR (0.46) NCEH1ARCA1CA2MAPT
SCHEMBL7335259 0.76 NCEH1 (0.43) NCEH1ARALDH1A1GAAPDE4A
SCHEMBL7344835 0.76 AR (0.36) NCEH1ARPDE4APDE4BPDE4C
SCHEMBL7344831 0.76 AR (0.36) NCEH1ARPDE4APDE4BPDE4C
Acetone SCHEMBL28054480 0.76 AR (0.57) CA9ARALDH1A1CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6358995-B1 AGONIST FOR RETINOIC ACID RECEPTORS; CAN BE SUBSTITUTED FOR RETINOIC ACID AS PREVENTIVE AND THERAPEUTIC DRUGS FOR VARIOUS DISEASES OR CANCERS, SUCH AS ACUTE PROMYELOCYTIC LEUKEMIA. EISAI CO., LTD. (JP) 2002-03-19 US disclosed
US-6121309-A SUCH AS 4-(2-(5-(7-FLUORO-4-TRIFLUOROMETHYLBENZOFURAN-2-YL)PYRROLYL)) BENZOIC ACID; RETINOIC ACID RECEPTOR AGONISM EISAI CO., LTD. (JP) 2000-09-19 US disclosed
US-6110959-A A RETINOIC ACID RECEPTOR AGONIST EISAI CO., LTD. (JP) 2000-08-29 US disclosed
EP-0889032-A1 FUSED-RING CARBOXYLIC ACID DERIVATIVES Eisai Co., Ltd. (JP) 1999-01-07 EP disclosed